Found 14 Enz. Inhib. hit(s) with Target = 'Prostaglandin G/H synthase 2' and Ligand = 'BDBM50174201'
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Affinity DataIC50: 800nMAssay Description:Inhibition of human recombinant COX2 by colorimetric analysisMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Affinity DataIC50: 800nMAssay Description:Inhibition of human recombinant COX2 catalytic activity using arachidonic acid as substrate pre-incubated for 10 mins followed by substrate addition ...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Affinity DataIC50: 800nMAssay Description:Inhibition of recombinant human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate by colorimetric methodMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Affinity DataIC50: 840nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Affinity DataIC50: 840nMAssay Description:Inhibition of human recombinant COX-2 using arachidonic acid as substrate preincubated with enzyme for 5 mins followed by substrate addition by color...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Dallas Department Of Veterans Affairs Medical Center
Curated by PDSP Ki Database
Affinity DataIC50: 840nMAssay Description:Inhibition of human recombinant COX2 using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition and measured after 2...More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of ovine COX2 assessed as PGF2alpha production from PGH2 after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of ovine COX2 by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair