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Found 2 Enz. Inhib. hit(s) with Target = 'Protein-glutamine gamma-glutamyltransferase 2' and Ligand = 'BDBM59177'
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59177(Dihydroisoxazole, 1e | Dihydroisoxazole, 1f)
Affinity DataKi:  1.10E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59177(Dihydroisoxazole, 1e | Dihydroisoxazole, 1f)
Affinity DataKi:  3.10E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed