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Found 1 Enz. Inhib. hit(s) with Target = 'Protein-glutamine gamma-glutamyltransferase E' and Ligand = 'BDBM577483'
TargetProtein-glutamine gamma-glutamyltransferase E(Homo sapiens (Human))
Zedira

US Patent
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  6.65E+4nMAssay Description:The most relevant off-targets are the transglutaminase isoenzymes especially tissue transglutaminase (TG2) because the enzyme is ubiquitously express...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent