Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 2' and Ligand = 'BDBM50329494'
TargetProteinase-activated receptor 2(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50329494(5-isoxazoyl-Cha-Ile-(3-aminophenyl)-(4-[aminomethy...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at PAR2 receptor in human HT-29 cells assessed as induction of intracellular calcium releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed