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Found 2 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 2' and Ligand = 'BDBM50440850'
TargetProteinase-activated receptor 2(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50440850(CHEMBL238396)
Affinity DataEC50:  220nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50440850(CHEMBL238396)
Affinity DataEC50:  100nMAssay Description:Agonist activity at PAR2 in human HT-29 cells assessed as increase in intracellular calcium releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed