Found 2 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 2' and Ligand = 'BDBM50440850'
TargetProteinase-activated receptor 2(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 220nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
TargetProteinase-activated receptor 2(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Agonist activity at PAR2 in human HT-29 cells assessed as increase in intracellular calcium releaseMore data for this Ligand-Target Pair