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Found 3 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 2' and Ligand = 'BDBM50503927'
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50503927(CHEMBL4470628)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at PAR2 in human EAhy926 cells assessed as inhibition of trypsin-induced intracellular calcium mobilization preincubated for 15 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50503927(CHEMBL4470628)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at PAR2 in human EAhy926 cells assessed as inhibition of SLIGKV-NH2-induced intracellular calcium mobilization preincubated for 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50503927(CHEMBL4470628)
Affinity DataIC50:  480nMAssay Description:Antagonist activity at PAR2 in human MDA-MB-231 cells assessed as inhibition of SLIGKV-NH2-induced intracellular calcium mobilization preincubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed