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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Chk1' and Ligand = 'BDBM50321677'
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50321677(6-phenyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazine...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of CHK1 by DELFIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50321677(6-phenyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazine...)
Affinity DataIC50:  5.89E+7nMAssay Description:Inhibition of CHK1 (unknown origin) assessed as inhibition of CDC25 phosphorylation after 30 min by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails Article