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Found 4 Enz. Inhib. hit(s) with Target = 'Short transient receptor potential channel 5' and Ligand = 'BDBM50529422'
TargetShort transient receptor potential channel 5(Homo sapiens (Human))
Goldfinch Bio

Curated by ChEMBL
LigandPNGBDBM50529422(CHEMBL4447753)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of (-)-Englerin-activated human TRPC5 channel expressed in HEK293 cells measured at holding potential of -60 mV by Q-patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetShort transient receptor potential channel 5(Homo sapiens (Human))
Goldfinch Bio

Curated by ChEMBL
LigandPNGBDBM50529422(CHEMBL4447753)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of lanthanum-activated human TRPC5 channel expressed in HEK293 cells measured at holding potential of -60 mV by Q-patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetShort transient receptor potential channel 5(Homo sapiens (Human))
Goldfinch Bio

Curated by ChEMBL
LigandPNGBDBM50529422(CHEMBL4447753)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetShort transient receptor potential channel 5(Homo sapiens (Human))
Goldfinch Bio

Curated by ChEMBL
LigandPNGBDBM50529422(CHEMBL4447753)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of riluzole-activated human TRPC5 channel expressed in HEK293 cells measured at holding potential of -60 mV by Q-patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed