Found 5 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50014407'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]-5HT from human SERTMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Ability to displace [3H]paroxetine bound to Serotonin transporter receptor in rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Binding affinity towards Serotonin transporter was determined in rat forebrain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Effect of compound on Serotonin transporter uptake from rat cortex using [3H]citalopram as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Inhibition of [3H]citalopram binding to Serotonin transporter of rat cerebral cortexMore data for this Ligand-Target Pair