Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with Target = 'Steryl-sulfatase' and Ligand = 'BDBM50118560'
TargetSteryl-sulfatase(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50118560(Sulfamic acid 2-adamantan-1-yl-4-oxo-4H-thiochrome...)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of recombinant human estrone sulfatase using 4-methylumbelliferyl sulfate as substrate by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2017
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50118560(Sulfamic acid 2-adamantan-1-yl-4-oxo-4H-thiochrome...)
Affinity DataIC50: 0.340nMAssay Description:Inhibitory activity against purified human steroid sulfatase (STS)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50118560(Sulfamic acid 2-adamantan-1-yl-4-oxo-4H-thiochrome...)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of steroid sulfataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50118560(Sulfamic acid 2-adamantan-1-yl-4-oxo-4H-thiochrome...)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of sulfatase (unknown origin) using 4-MUS as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50118560(Sulfamic acid 2-adamantan-1-yl-4-oxo-4H-thiochrome...)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of human steroid sulfatase by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50118560(Sulfamic acid 2-adamantan-1-yl-4-oxo-4H-thiochrome...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against human steroid sulfatase over-expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50118560(Sulfamic acid 2-adamantan-1-yl-4-oxo-4H-thiochrome...)
Affinity DataKi:  210nMAssay Description:Inhibitory activity against human steroid sulfataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed