Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with Target = 'Steryl-sulfatase' and Ligand = 'BDBM50266402'
TargetSteryl-sulfatase(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50266402(CHEMBL4071245)
Affinity DataIC50: 15nMAssay Description:Inhibition of human STS expressed in human T47D cells using [3H]E1S as substrate incubated for 1 hr followed by substrate addition measured after 24 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSteryl-sulfatase(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50266402(CHEMBL4071245)
Affinity DataIC50: 16nMAssay Description:Inhibition of STS in human T47D cells preincubated for 1 hr followed by addition of [3H]-E1S/E1S as substrate measured after 24 hrs by HPLC based rad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSteryl-sulfatase(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50266402(CHEMBL4071245)
Affinity DataIC50: 16nMAssay Description:Irreversible inhibition of STS in human T47D cells preincubated for 2 hrs followed by compound washout and addition of [3H]-E1S/E1S as substrate meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSteryl-sulfatase(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50266402(CHEMBL4071245)
Affinity DataIC50: 16nMAssay Description:Irreversible inhibition of human STS expressed in human T47D cells using [3H]E1S as substrate preincubated for 2 hr followed by substrate addition me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSteryl-sulfatase(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50266402(CHEMBL4071245)
Affinity DataIC50: 143nMAssay Description:Inhibition of human placental microsomal STS assessed as formation of E1 preincubated for 30 mins followed by addition of E1S as substrate measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed