TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.780nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.05nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 53nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 53.1nMAssay Description:Activity at TPbeta (long isoform) receptor expressed in HEK293 cells assessed as ability to antagonize U46619-mediated calcium ion mobilizationMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 240nMAssay Description:Inhibition of U46619-induced platelet aggregationMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 319nMAssay Description:Activity at TPalpha (short isoform) receptor expressed in HEK293 cells assessed as ability to antagonize U46619-mediated calcium ion mobilizationMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 319nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 620nMAssay Description:Antagonist activity at human thromboxane A2 receptor beta over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular calc...More data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 700nMAssay Description:Antagonist activity at human thromboxane A2 receptor alpha over-expressed in HEK293 cells assessed as inhibition of U-46619-induced intracellular cal...More data for this Ligand-Target Pair