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Found 6 Enz. Inhib. hit(s) with Target = 'Trace amine-associated receptor 1' and Ligand = 'BDBM50336205'
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336205((N-(3-Ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoro...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336205((N-(3-Ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoro...)
Affinity DataKi:  942nMAssay Description:Inhibition of rat TAAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336205((N-(3-Ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoro...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human TAAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336205((N-(3-Ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoro...)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336205((N-(3-Ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoro...)
Affinity DataIC50:  4.54E+3nMAssay Description:Antagonist activity at rat TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336205((N-(3-Ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoro...)
Affinity DataIC50:  7.49E+3nMAssay Description:Antagonist activity at human TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed