Report error Found 5 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM22988'
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale
Universita Del Piemonte Orientale
Affinity DataEC50: 200nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale
Universita Del Piemonte Orientale
Affinity DataEC50: 630nMAssay Description:Activation of human VR1 expressed in HEK293 cells assessed as stimulation of Ca2+ influxMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale
Universita Del Piemonte Orientale
Affinity DataEC50: 490nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale
Universita Del Piemonte Orientale
Affinity DataEC50: 16nMAssay Description:Agonist activity at TRPV1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Universidad Complutense
Curated by ChEMBL
Universidad Complutense
Curated by ChEMBL
Affinity DataKi: 169nMAssay Description:Binding affinity to vanilloid VR1 receptor using [3H]resiniferatoxin ([3H]-RTX) in rat spinal cord membranesMore data for this Ligand-Target Pair
