Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM50285610'
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluorescence as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV1 (unknown origin) activationMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataIC50: 1.19E+4nMAssay Description:Agonist activity at ionomycin-stimulated TRPV1 (unknown origin) channel desensitization in presence of capsaicinMore data for this Ligand-Target Pair
In DepthDetails
PubMed