Report error Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 4' and Ligand = 'BDBM50463445'
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataEC50: 3.30E+3nMAssay Description:Agonist activity at rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of GSK1016790A-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
