Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor' and Ligand = 'BDBM50038189'
TargetType-1 angiotensin II receptor(Rabbit)
The M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataKd:  0.0501nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
The M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataIC50: 0.200nMAssay Description:In vitro binding affinity for angiotensin II AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
The M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataIC50: 0.200nMAssay Description:Compound was evaluated for inhibition of 125I[Sar1,Ile8] all binding to rabbit aorta Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
The M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity was evaluated against Angiotensin II receptor, type 1 in rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at angiotensin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
The M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataIC50: 0.200nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
The M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Angiotensin II receptor type 1 in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article