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Found 4 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor A/B' and Ligand = 'BDBM50228308'
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228308(CHEMBL413740)
Affinity DataIC50:  0.900nMAssay Description:Inhibitory concentration against [125 I]Ang II binding to rat pituitary membranes Angiotensin II receptor type 1 without 0.2% bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228308(CHEMBL413740)
Affinity DataIC50:  2.60nMAssay Description:Concentration required to 50% inhibition in specific binding of [125- I]A-II to Angiotensin II receptor in rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228308(CHEMBL413740)
Affinity DataIC50:  2.60nMAssay Description:Inhibitory concentration against specific binding of [125 I]Ang II to rat uterine membranes (Angiotensin II receptor, type 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228308(CHEMBL413740)
Affinity DataIC50:  3.80nMAssay Description:Inhibitory concentration against specific binding of [125 I]Ang II to rat pituitary membranes (Angiotensin II receptor, type 1) in presence of 0.2% b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed