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Report error Found 4 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ABL1' and Ligand = 'BDBM50320700'
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Institute of Molecular Genetics Igm-Cnr

Curated by ChEMBL
LigandPNGBDBM50320700(1-[2-chloro-2-(4-fluorophenyl)ethyl]-N-(3-fluoroph...)
Affinity DataKi:  700nMAssay Description:Inhibition of histidine-tagged human recombinant ABL expressed in baculovirus system assessed as [gamma32P]ATP utilization after 10 mins by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Institute of Molecular Genetics Igm-Cnr

Curated by ChEMBL
LigandPNGBDBM50320700(1-[2-chloro-2-(4-fluorophenyl)ethyl]-N-(3-fluoroph...)
Affinity DataKi:  732nMAssay Description:Binding affinity to recombinant wild type human Abl using abitide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Institute of Molecular Genetics Igm-Cnr

Curated by ChEMBL
LigandPNGBDBM50320700(1-[2-chloro-2-(4-fluorophenyl)ethyl]-N-(3-fluoroph...)
Affinity DataKi:  750nMAssay Description:Inhibition of histidine-tagged human recombinant ABL expressed in baculovirus system assessed as [gamma32P]ATP utilization after 10 mins by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Institute of Molecular Genetics Igm-Cnr

Curated by ChEMBL
LigandPNGBDBM50320700(1-[2-chloro-2-(4-fluorophenyl)ethyl]-N-(3-fluoroph...)
Affinity DataKi:  3.00E+3nMAssay Description:Mixed-type inhibition of histidine-tagged human recombinant ABL expressed in baculovirus system assessed as [gamma32P]ATP utilization after 10 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed