Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase Lck' and Ligand = 'BDBM50111444'
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50111444(2-{4-[2-[1-(4-Methoxy-benzyl)-4-methyl-2-oxo-1,2-d...)
Affinity DataKd:  1.00E+3nMAssay Description:Inhibition of p56 Lck SH2 domain binding to pYEEIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50111444(2-{4-[2-[1-(4-Methoxy-benzyl)-4-methyl-2-oxo-1,2-d...)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of calcium release in Jurkat cells after T-cell receptor cross linking antibody treatmentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50111444(2-{4-[2-[1-(4-Methoxy-benzyl)-4-methyl-2-oxo-1,2-d...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity for p56lck SH2 domain siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50111444(2-{4-[2-[1-(4-Methoxy-benzyl)-4-methyl-2-oxo-1,2-d...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity for p56 lck kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed