Report error Found 8 Enz. Inhib. hit(s) with Target = 'Vascular endothelial growth factor receptor 1' and Ligand = 'BDBM4814'
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal GST-tagged Flt1 using poly(Glu,Tyr) as substrate after 60 mins by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Binding affinity to FLT1More data for this Ligand-Target Pair
Affinity DataKd: 1.80nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Binding constant for FLT1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Binding constant for FLT1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to VEGFR1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant GST-fused VEGFR1 kinase domain transphosphorylation expressed in baculovirus expression system using poly-Glu-Tyr (4:...More data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:Inhibition of VEGFR1 (unknown origin) incubated for 30 mins in presence of ATP by mobility shift assayMore data for this Ligand-Target Pair
