Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM50307117'
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50307117(N-(4-(2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carb...)
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at V1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50307117(N-(4-(2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carb...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50307117(N-(4-(2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carb...)
Affinity DataKi:  2.74nMAssay Description:Displacement of [3H]-AVP from human vasopressin V1a receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50307117(N-(4-(2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carb...)
Affinity DataKi:  2.74nMAssay Description:Displacement of [3H]AVP from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50307117(N-(4-(2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carb...)
Affinity DataEC50:  14nMAssay Description:Activity at human vasopressin V1a receptor expressed in CHO cells by NFAT-luciferase gene reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50307117(N-(4-(2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carb...)
Affinity DataKi:  14.1nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed