Affinity DataKi: 0.650nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Binding affinity to human vasopressin V1b receptor expressed CHO cells after 1 hr by spectrofluorimetry analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 2.48nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed CHO cells assessed as induction of phospholipase C activity after 15 mins by inositol ph...More data for this Ligand-Target Pair