Found 9 Enz. Inhib. hit(s) with Target = 'Vasopressin V2 receptor' and Ligand = 'BDBM35723' TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Affinity DataKi: 0.430nMAssay Description:Concentration of the compound which inhibit [3H]-AVP binding to human Vasopressin V2 receptor coded HeLa cells by 50%More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V2 receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindin...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Affinity DataKi: 1.70nMAssay Description:Displacement of conivaptan-red from SNAP-tagged V2 receptor (unknown origin) expressed in HEK293 cells assessed as inhibition constant measured after...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Affinity DataKi: 2.40nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Affinity DataIC50: 0.00700nMAssay Description:Antagonist activity at human AVPR2 by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Affinity DataIC50: 3nMpH: 7.4 T: 2°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human V2 receptor expressed in CHO cells assessed as reduction in vasopressin induced cAMP production preincubated for 30 mins...More data for this Ligand-Target Pair
