Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Vitamin D3 receptor' and Ligand = 'BDBM50397222'
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50397222(CHEMBL2172538)
Affinity DataIC50:  27.3nMAssay Description:Binding affinity to VDR assessed as inhibition of fluorescent ligand by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50397222(CHEMBL2172538)
Affinity DataEC50:  9.04nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed