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TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKd:  6.30nMAssay Description:Displacement of [3H]epibatidine from chimeric human alpha7-5-HT3A receptor expressed in HEK293 cells after 2 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50353944(CHEMBL1831036)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology assa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50353945(CHEMBL1831033)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology assa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50353946(CHEMBL1831032)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology assa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50353947(CHEMBL1831030)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology assa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50353948(CHEMBL1831043)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology assa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50353949(CHEMBL1831038)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology assa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419175(CHEMBL1831034)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419184(CHEMBL1831046)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419182(CHEMBL1831044)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419181(CHEMBL1831042)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419179(CHEMBL1831035)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50485643(3-Phenylquinuclidine | CHEMBL1890808)
Affinity DataIC50: 200nMAssay Description:Displacement of [3H]epibatidine from chimeric human alpha7-5-HT3A receptor expressed in HEK293 cells after 2 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50267844(3-(10,11-Dihydro-5H-dibenzo[a,d]cyclohepten-5-ylox...)
Affinity DataIC50: 210nMAssay Description:Activity at human alpha4beta2 nAChR expressed in Xenopus oocytes assessed as inhibition of acetylcholine-evoked currentMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50485639(CHEMBL2147673)
Affinity DataIC50: 400nMAssay Description:Displacement of [3H]epibatidine from chimeric human alpha7-5-HT3A receptor expressed in HEK293 cells after 2 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50267883(8-Benzyl-3-(10,11-dihydro-5H-dibenzo[a,d]cyclohept...)
Affinity DataIC50: 460nMAssay Description:Activity at human alpha4beta2 nAChR expressed in Xenopus oocytes assessed as inhibition of acetylcholine-evoked currentMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50267844(3-(10,11-Dihydro-5H-dibenzo[a,d]cyclohepten-5-ylox...)
Affinity DataIC50: 880nMAssay Description:Activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as inhibition of acetylcholine-evoked currentMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50267883(8-Benzyl-3-(10,11-dihydro-5H-dibenzo[a,d]cyclohept...)
Affinity DataIC50: 1.73E+3nMAssay Description:Activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as inhibition of acetylcholine-evoked currentMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 12(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492460(CHEMBL2402776)
Affinity DataKi:  0.240nMAssay Description:Inhibition of human recombinant carbonic anhydrase 12 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492476(CHEMBL1518649)
Affinity DataKi:  0.25nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492471(CHEMBL2402764)
Affinity DataKi:  0.310nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492464(CHEMBL2402768)
Affinity DataKi:  0.320nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492460(CHEMBL2402776)
Affinity DataKi:  0.410nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 12(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492476(CHEMBL1518649)
Affinity DataKi:  0.430nMAssay Description:Inhibition of human recombinant carbonic anhydrase 12 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492465(CHEMBL2402767)
Affinity DataKi:  0.440nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492477(CHEMBL2402758)
Affinity DataKi:  0.450nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492474(CHEMBL2402753)
Affinity DataKi:  0.520nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492467(CHEMBL2402756)
Affinity DataKi:  0.530nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 12(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492481(CHEMBL2402754)
Affinity DataKi:  0.540nMAssay Description:Inhibition of human recombinant carbonic anhydrase 12 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492456(CHEMBL2402760)
Affinity DataKi:  0.570nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 12(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492467(CHEMBL2402756)
Affinity DataKi:  0.570nMAssay Description:Inhibition of human recombinant carbonic anhydrase 12 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492454(CHEMBL2402763)
Affinity DataKi:  0.610nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492481(CHEMBL2402754)
Affinity DataKi:  0.620nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 12(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492470(CHEMBL2402771)
Affinity DataKi:  0.620nMAssay Description:Inhibition of human recombinant carbonic anhydrase 12 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 12(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492471(CHEMBL2402764)
Affinity DataKi:  0.630nMAssay Description:Inhibition of human recombinant carbonic anhydrase 12 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 12(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492464(CHEMBL2402768)
Affinity DataKi:  0.640nMAssay Description:Inhibition of human recombinant carbonic anhydrase 12 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492481(CHEMBL2402754)
Affinity DataKi:  0.690nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins to 6 hrs by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492481(CHEMBL2402754)
Affinity DataKi:  0.690nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492454(CHEMBL2402763)
Affinity DataKi:  0.700nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins to 6 hrs by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492455(CHEMBL2402762)
Affinity DataKi:  0.700nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins to 6 hrs by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492455(CHEMBL2402762)
Affinity DataKi:  0.700nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492454(CHEMBL2402763)
Affinity DataKi:  0.700nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492456(CHEMBL2402760)
Affinity DataKi:  0.720nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins to 6 hrs by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492456(CHEMBL2402760)
Affinity DataKi:  0.720nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492460(CHEMBL2402776)
Affinity DataKi:  0.740nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins to 6 hrs by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492460(CHEMBL2402776)
Affinity DataKi:  0.740nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 12(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492454(CHEMBL2402763)
Affinity DataKi:  0.740nMAssay Description:Inhibition of human recombinant carbonic anhydrase 12 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50492461(CHEMBL2402775)
Affinity DataKi:  0.740nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492471(CHEMBL2402764)
Affinity DataKi:  0.760nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins to 6 hrs by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50492471(CHEMBL2402764)
Affinity DataKi:  0.760nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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