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Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245828(2-Tosylnaphthalene-1,4-diol | CHEMBL509952)
Affinity DataIC50:  0.610nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245923(2-(naphthalen-2-ylsulfonyl)naphthalene-1,4-diol | ...)
Affinity DataIC50:  1.49nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245928(2-tosylnaphthalene-1,4-dione | CHEMBL454282)
Affinity DataIC50:  1.99nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245877(2-(phenylsulfonyl)naphthalene-1,4-diol | CHEMBL462...)
Affinity DataIC50:  2.84nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245880(2-(4-propylphenylsulfonyl)naphthalene-1,4-diol | C...)
Affinity DataIC50:  3.09nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245830(3-(1,4-dihydroxynaphthalen-2-ylsulfonyl)propanoic ...)
Affinity DataIC50:  3.53nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245829(2-(methylsulfonyl)naphthalene-1,4-diol | CHEMBL491...)
Affinity DataIC50:  3.53nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245879(2-(4-chlorophenylsulfonyl)naphthalene-1,4-diol | C...)
Affinity DataIC50:  3.61nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245878(CHEMBL512926 | N-(4-(1,4-dihydroxynaphthalen-2-yls...)
Affinity DataIC50:  3.76nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245924(2-tosylanthracene-1,4-diol | CHEMBL451059)
Affinity DataIC50:  8.47nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-ketoacyl-[acyl-carrier-protein] synthase III(malaria parasite P. falciparum)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245829(2-(methylsulfonyl)naphthalene-1,4-diol | CHEMBL491...)
Affinity DataIC50:  27.4nMAssay Description:Inhibition of Plasmodium falciparum FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-ketoacyl-[acyl-carrier-protein] synthase III(malaria parasite P. falciparum)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245878(CHEMBL512926 | N-(4-(1,4-dihydroxynaphthalen-2-yls...)
Affinity DataIC50:  29.6nMAssay Description:Inhibition of Plasmodium falciparum FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245926(CHEMBL462376 | N-(4-(2,5-dihydroxyphenylsulfonyl)p...)
Affinity DataIC50:  31.4nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245925(2-tosylbenzene-1,4-diol | CHEMBL462375)
Affinity DataIC50:  34.4nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-ketoacyl-[acyl-carrier-protein] synthase III(malaria parasite P. falciparum)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245830(3-(1,4-dihydroxynaphthalen-2-ylsulfonyl)propanoic ...)
Affinity DataIC50:  46.5nMAssay Description:Inhibition of Plasmodium falciparum FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-ketoacyl-[acyl-carrier-protein] synthase III(malaria parasite P. falciparum)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245880(2-(4-propylphenylsulfonyl)naphthalene-1,4-diol | C...)
Affinity DataIC50:  72.6nMAssay Description:Inhibition of Plasmodium falciparum FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-ketoacyl-[acyl-carrier-protein] synthase III(malaria parasite P. falciparum)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245828(2-Tosylnaphthalene-1,4-diol | CHEMBL509952)
Affinity DataIC50:  73.6nMAssay Description:Inhibition of Plasmodium falciparum FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245831(2-(p-tolylthio)naphthalene-1,4-dione | CHEMBL50155...)
Affinity DataIC50:  112nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-ketoacyl-[acyl-carrier-protein] synthase III(malaria parasite P. falciparum)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245879(2-(4-chlorophenylsulfonyl)naphthalene-1,4-diol | C...)
Affinity DataIC50:  129nMAssay Description:Inhibition of Plasmodium falciparum FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245927(2-tosylnaphthalene | CHEMBL462553)
Affinity DataIC50:  138nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138357(US10278929, Compound 6 | US11337935, Compound 6 | ...)
Affinity DataIC50:  277nMAssay Description:Table 3: The FP assay was then adapted for HTS and used to screen 120,000 small molecule library for compounds that displaced probe 5 from the T4 bin...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138357(US10278929, Compound 6 | US11337935, Compound 6 | ...)
Affinity DataIC50:  277nMAssay Description:The FP assay was then adapted for HTS and used to screen a ˜120,000 member small molecule library for compounds that displaced the FP probe from the ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138357(US10278929, Compound 6 | US11337935, Compound 6 | ...)
Affinity DataIC50:  277nMAssay Description:The FP assay was then adapted for HTS and used to screen ~120,000 small molecule library for compounds that displaced probe 5 from the T4 binding of ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetBeta-ketoacyl-[acyl-carrier-protein] synthase III(malaria parasite P. falciparum)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245877(2-(phenylsulfonyl)naphthalene-1,4-diol | CHEMBL462...)
Affinity DataIC50:  279nMAssay Description:Inhibition of Plasmodium falciparum FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM85507(CAS_4394-00-7 | NSC_4488 | Niflumic acid | Niflumi...)
Affinity DataIC50:  289nMAssay Description:Table 3: The FP assay was then adapted for HTS and used to screen 120,000 small molecule library for compounds that displaced probe 5 from the T4 bin...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM85507(CAS_4394-00-7 | NSC_4488 | Niflumic acid | Niflumi...)
Affinity DataIC50:  289nMAssay Description:The FP assay was then adapted for HTS and used to screen ~120,000 small molecule library for compounds that displaced probe 5 from the T4 binding of ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM85507(CAS_4394-00-7 | NSC_4488 | Niflumic acid | Niflumi...)
Affinity DataIC50:  289nMAssay Description:The FP assay was then adapted for HTS and used to screen a ˜120,000 member small molecule library for compounds that displaced the FP probe from the ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138358(US10278929, Compound 7 | US11337935, Compound 7 | ...)
Affinity DataIC50:  296nMAssay Description:Table 3: The FP assay was then adapted for HTS and used to screen 120,000 small molecule library for compounds that displaced probe 5 from the T4 bin...More data for this Ligand-Target Pair
TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138358(US10278929, Compound 7 | US11337935, Compound 7 | ...)
Affinity DataIC50:  296nMAssay Description:The FP assay was then adapted for HTS and used to screen a ˜120,000 member small molecule library for compounds that displaced the FP probe from the ...More data for this Ligand-Target Pair
TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138358(US10278929, Compound 7 | US11337935, Compound 7 | ...)
Affinity DataIC50:  296nMAssay Description:The FP assay was then adapted for HTS and used to screen ~120,000 small molecule library for compounds that displaced probe 5 from the T4 binding of ...More data for this Ligand-Target Pair
TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM50308343((Z)-5-(3,5-dibromo-4-methoxybenzylidene)thiazolidi...)
Affinity DataIC50:  301nMAssay Description:Table 3: The FP assay was then adapted for HTS and used to screen 120,000 small molecule library for compounds that displaced probe 5 from the T4 bin...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM50308343((Z)-5-(3,5-dibromo-4-methoxybenzylidene)thiazolidi...)
Affinity DataIC50:  301nMAssay Description:The FP assay was then adapted for HTS and used to screen ~120,000 small molecule library for compounds that displaced probe 5 from the T4 binding of ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM50308343((Z)-5-(3,5-dibromo-4-methoxybenzylidene)thiazolidi...)
Affinity DataIC50:  301nMAssay Description:The FP assay was then adapted for HTS and used to screen a ˜120,000 member small molecule library for compounds that displaced the FP probe from the ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138359(US10278929, Compound 9 | US11337935, Compound 9 | ...)
Affinity DataIC50:  329nMAssay Description:Table 3: The FP assay was then adapted for HTS and used to screen 120,000 small molecule library for compounds that displaced probe 5 from the T4 bin...More data for this Ligand-Target Pair
TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138359(US10278929, Compound 9 | US11337935, Compound 9 | ...)
Affinity DataIC50:  329nMAssay Description:The FP assay was then adapted for HTS and used to screen a ˜120,000 member small molecule library for compounds that displaced the FP probe from the ...More data for this Ligand-Target Pair
TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138359(US10278929, Compound 9 | US11337935, Compound 9 | ...)
Affinity DataIC50:  329nMAssay Description:The FP assay was then adapted for HTS and used to screen ~120,000 small molecule library for compounds that displaced probe 5 from the T4 binding of ...More data for this Ligand-Target Pair
TargetBeta-ketoacyl-[acyl-carrier-protein] synthase III(malaria parasite P. falciparum)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245924(2-tosylanthracene-1,4-diol | CHEMBL451059)
Affinity DataIC50:  341nMAssay Description:Inhibition of Plasmodium falciparum FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-ketoacyl-[acyl-carrier-protein] synthase III(malaria parasite P. falciparum)
Portland State University

Curated by ChEMBL
LigandPNGBDBM50245923(2-(naphthalen-2-ylsulfonyl)naphthalene-1,4-diol | ...)
Affinity DataIC50:  393nMAssay Description:Inhibition of Plasmodium falciparum FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138360(US10278929, Compound 10 | US11337935, Compound 10 ...)
Affinity DataIC50:  433nMAssay Description:Table 3: The FP assay was then adapted for HTS and used to screen 120,000 small molecule library for compounds that displaced probe 5 from the T4 bin...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138360(US10278929, Compound 10 | US11337935, Compound 10 ...)
Affinity DataIC50:  433nMAssay Description:The FP assay was then adapted for HTS and used to screen a ˜120,000 member small molecule library for compounds that displaced the FP probe from the ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138360(US10278929, Compound 10 | US11337935, Compound 10 ...)
Affinity DataIC50:  433nMAssay Description:The FP assay was then adapted for HTS and used to screen ~120,000 small molecule library for compounds that displaced probe 5 from the T4 binding of ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM22971(2-[(2,6-dichloro-3-methylphenyl)amino]benzoic acid...)
Affinity DataIC50:  504nMAssay Description:Table 3: The FP assay was then adapted for HTS and used to screen 120,000 small molecule library for compounds that displaced probe 5 from the T4 bin...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138361(US8877795, Meclofenamic Acid)
Affinity DataIC50:  504nMAssay Description:The FP assay was then adapted for HTS and used to screen ~120,000 small molecule library for compounds that displaced probe 5 from the T4 binding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM383181(US10278929, Meclofenamic acid)
Affinity DataIC50:  504nMAssay Description:The FP assay was then adapted for HTS and used to screen a ˜120,000 member small molecule library for compounds that displaced the FP probe from the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM138362(US8877795, 11)
Affinity DataIC50:  586nMAssay Description:The FP assay was then adapted for HTS and used to screen ~120,000 small molecule library for compounds that displaced probe 5 from the T4 binding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM58032(2-(1,3-Dioxo-indan-2-yl)-2-(2-methyl-1H-indol-3-yl...)
Affinity DataIC50:  586nMAssay Description:The FP assay was then adapted for HTS and used to screen a ˜120,000 member small molecule library for compounds that displaced the FP probe from the ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM554486(US11337935, Compound 11)
Affinity DataIC50:  586nMAssay Description:Table 3: The FP assay was then adapted for HTS and used to screen 120,000 small molecule library for compounds that displaced probe 5 from the T4 bin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  653nMAssay Description:Table 3: The FP assay was then adapted for HTS and used to screen 120,000 small molecule library for compounds that displaced probe 5 from the T4 bin...More data for this Ligand-Target Pair
TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  653nMAssay Description:The FP assay was then adapted for HTS and used to screen a ˜120,000 member small molecule library for compounds that displaced the FP probe from the ...More data for this Ligand-Target Pair
TargetTransthyretin(Human)
Leland Stanford Junior University

US Patent
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  653nMAssay Description:The FP assay was then adapted for HTS and used to screen ~120,000 small molecule library for compounds that displaced probe 5 from the T4 binding of ...More data for this Ligand-Target Pair
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