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TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504252(CHEMBL3098650)
Affinity DataIC50: 38nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50537171(CHEMBL4576947)
Affinity DataIC50: 40nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504264(CHEMBL4561572)
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50537172(CHEMBL4520252)
Affinity DataIC50: 41nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Cairo University

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 41nMAssay Description:Inhibition of ovine COX-1 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 49nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L3(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50431630(KRX-0401 | PERIFOSINE)
Affinity DataIC50: 50nMAssay Description:Inhibition of UCHL3 (unknown origin) assessed as reduction in RAD51 deubiquitination incubated for 4 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504265(CHEMBL4529762)
Affinity DataIC50: 53nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504267(CHEMBL4465282)
Affinity DataIC50: 59nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504253(CHEMBL1322701)
Affinity DataIC50: 63nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504255(CHEMBL3098648)
Affinity DataIC50: 69nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50571800(CHEMBL4871569)
Affinity DataIC50: 72nMAssay Description:Inhibition of autophosphorylation of EGFR (unknown origin) by Cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504251(CHEMBL4541315)
Affinity DataIC50: 81nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 87nMAssay Description:Inhibition of autophosphorylation of EGFR (unknown origin) by Cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504256(CHEMBL4450458)
Affinity DataIC50: 89nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504263(CHEMBL4475508)
Affinity DataIC50: 94nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504269(CHEMBL4576864)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504270(CHEMBL4456191)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504272(CHEMBL4444316)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504261(CHEMBL4440531)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504254(CHEMBL4569755)
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504268(CHEMBL4449489)
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504257(CHEMBL4535881)
Affinity DataIC50: 170nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504259(CHEMBL4573875)
Affinity DataIC50: 210nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Institut Pasteur

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataIC50: 220nMAssay Description:Inhibition of SARS-CoV-2 nsp14 guanine-N7-methyltransferase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L1(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50594734(CHEMBL5191704)
Affinity DataIC50: 230nMAssay Description:Inhibition of UCHL1 (unknown origin) using Ub-Rho-morpholine as substrate preincubated for 30 mins followed by substrate addition by fluorescence bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504260(CHEMBL4464158)
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50504257(CHEMBL4535881)
Affinity DataIC50: 276nMAssay Description:Inhibition of recombinant human GST-tagged EGFR catalytic domain (668 to 1210 residues) expressed in baculovirus expression system using TK-biotin pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504271(CHEMBL4450095)
Affinity DataIC50: 290nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504266(CHEMBL4462267)
Affinity DataIC50: 290nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504262(CHEMBL4571917)
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504250(CHEMBL4533452)
Affinity DataIC50: 380nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50504264(CHEMBL4561572)
Affinity DataIC50: 412nMAssay Description:Inhibition of recombinant human GST-tagged EGFR catalytic domain (668 to 1210 residues) expressed in baculovirus expression system using TK-biotin pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 418nMAssay Description:Inhibition of recombinant human GST-tagged EGFR catalytic domain (668 to 1210 residues) expressed in baculovirus expression system using TK-biotin pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504249(CHEMBL4571604)
Affinity DataIC50: 430nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50045333(CHEBI:90705 | SB-203580)
Affinity DataIC50: 500nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 510nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504258(CHEMBL4582518)
Affinity DataIC50: 560nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L3(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50594731(CHEMBL1241028)
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human UCHL3 expressed in baculovirus infected Sf9 cells using ubiquitin-AMC as substrate preincubated for 30 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L1(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50594736(CHEMBL5175498)
Affinity DataIC50: 670nMAssay Description:Inhibition of UCHL1 (unknown origin) using Ub-Rho as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetProstaglandin G/H synthase 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50174201(ARTHROTEC | GP 45840 | SOLARAZE | Sodium; [2-(2,6-...)
Affinity DataIC50: 840nMAssay Description:Inhibition of human recombinant COX-2 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50504254(CHEMBL4569755)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR catalytic domain (668 to 1210 residues) expressed in baculovirus expression system using TK-biotin pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L3(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50069764(CHEMBL3407501)
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of UCHL3 (unknown origin) using ubiquitin-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50174201(ARTHROTEC | GP 45840 | SOLARAZE | Sodium; [2-(2,6-...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of ovine COX-1 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504265(CHEMBL4529762)
Affinity DataIC50: 4.17E+3nMAssay Description:Inhibition of ovine COX-1 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504252(CHEMBL3098650)
Affinity DataIC50: 4.49E+3nMAssay Description:Inhibition of ovine COX-1 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L3(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50594730(CHEMBL5193983)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of UCHL3 (unknown origin) incubated for 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504267(CHEMBL4465282)
Affinity DataIC50: 5.39E+3nMAssay Description:Inhibition of ovine COX-1 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50504272(CHEMBL4444316)
Affinity DataIC50: 5.71E+3nMAssay Description:Inhibition of ovine COX-1 by EIA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L1(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50594735(CHEMBL5185124)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of UCHL1 (unknown origin) using Ub-Rho as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
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