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TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039675(3-[(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-p...)
Affinity DataKd:  0.690nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039674(Bromo-acetic acid 3-(2,6-dioxo-1,3-dipropyl-2,3,6,...)
Affinity DataKd:  0.710nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039678(8-cyclopentyl-1,3-di[3-(4-fluorosulfonylphenylcarb...)
Affinity DataKd:  0.820nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039696(3-Fluorosulfonyl-benzoic acid 3-(2,6-dioxo-1,3-dip...)
Affinity DataKd:  1.30nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039677(4-[3-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKd:  1.80nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039697(Bromo-acetic acid 2-(8-cyclopentyl-2,6-dioxo-1-pro...)
Affinity DataKd:  1.10nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039680(8-(2,5-Dioxo-2,5-dihydro-pyrrol-1-ylmethyl)-1,3-di...)
Affinity DataKd:  0.730nMAssay Description:Binding of [3H]-CPX to A1 adenosine receptor of DDT1 MF-2 (DDT) cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039684(2-Bromo-N-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahyd...)
Affinity DataKd:  1.30nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039689(3-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKd:  0.790nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039685(3-[2-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKd:  1.10nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039691(3-[3-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKd:  0.860nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039695(Bromo-acetic acid 3-(8-cyclopentyl-2,6-dioxo-1-pro...)
Affinity DataKd:  1.5nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039688(4-[2-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H...)
Affinity DataKd:  0.740nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039675(3-[(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-p...)
Affinity DataKd:  0.690nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039682(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKd:  1.10nMAssay Description:Specific binding of [3H]CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Deakin University

Curated by ChEMBL
LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.340nMAssay Description:Dissociation constant of [3H]ZM-241385 binding to adenosine A2A receptor(AR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.280nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 0.05 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A2a(Rat)
Deakin University

Curated by ChEMBL
LigandPNGBDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.230nMAssay Description:Dissociation constant of [3H]ZM-241385 binding to adenosine A2A receptor(AR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.360nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor(AR) at 5 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.330nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 5 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095603(4-[5-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.810nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.310nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 100 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.340nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 100 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.710nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 100 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.270nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 0.1 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095606(4-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetrahy...)
Affinity DataKd:  0.320nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.260nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 0.05 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.370nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 5 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095605(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.370nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.240nMAssay Description:Dissociation constant of [3H]DPCPX binding to adenosine A1 receptor(AR) at 0.1 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Deakin University

Curated by ChEMBL
LigandPNGBDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.270nMAssay Description:Dissociation constant of [3H]ZM-241385 binding to adenosine A2A receptor(AR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.360nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.360nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50120221(4-[5-(8-Bicyclo[2.2.1]hept-2-yl-2,6-dioxo-1-propyl...)
Affinity DataKd:  0.530nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50120223(4-[5-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.400nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.330nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.330nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50120223(4-[5-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.400nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50120221(4-[5-(8-Bicyclo[2.2.1]hept-2-yl-2,6-dioxo-1-propyl...)
Affinity DataKd:  0.530nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50120222(4-[5-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.530nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50120222(4-[5-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.530nMAssay Description:Equilibrium dissociation constant for [3H]DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50451007(CHEMBL2112106)
Affinity DataEC50:  1.10nMAssay Description:Adenosine receptor agonistic activity against isoproterenol (1 uM) stimulated cAMP accumulation in DDT MF-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50451006(CHEMBL2112185)
Affinity DataEC50:  1nMAssay Description:Adenosine receptor agonistic activity against isoproterenol (1 uM) stimulated cAMP accumulation in DDT MF-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50366624(CHEMBL608777 | CHEMBL3144085)
Affinity DataEC50:  7.10nMAssay Description:Adenosine receptor agonistic activity against isoproterenol (1 uM) stimulated cAMP accumulation in DDT MF-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50366625(CHEMBL608220)
Affinity DataEC50:  22nMAssay Description:Adenosine receptor agonistic activity against isoproterenol (1 uM) stimulated cAMP accumulation in DDT MF-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50366627(CHEMBL608223 | CHEMBL3144087)
Affinity DataEC50:  2.70nMAssay Description:Adenosine receptor agonistic activity against isoproterenol (1 uM) stimulated cAMP accumulation in DDT MF-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50366629(CHEMBL609070 | CHEMBL3144086)
Affinity DataEC50:  8nMAssay Description:Adenosine receptor agonistic activity against isoproterenol (1 uM) stimulated cAMP accumulation in DDT MF-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50366630(CHEMBL608219)
Affinity DataEC50:  9.20nMAssay Description:Adenosine receptor agonistic activity against isoproterenol (1 uM) stimulated cAMP accumulation in DDT MF-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50375517(CHEMBL411245)
Affinity DataIC50: 0.120nMAssay Description:Agonist activity at adenosine A1 receptor assessed as inhibition of isoproterenol-stimulated cAMP accumulation in DDT1MF-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50375516(CHEMBL258759)
Affinity DataIC50: 0.300nMAssay Description:Agonist activity at adenosine A1 receptor assessed as inhibition of isoproterenol-stimulated cAMP accumulation in DDT1MF-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
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