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LigandPNGBDBM24184((3-aminopropyl)phosphinic acid | CHEMBL112203 | CG...)
Affinity DataIC50: 5nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM24185(CGP35024 | 3-Apmpa | CHEMBL112710 | (3-aminopropyl...)
Affinity DataIC50: 16nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50033007((3-Amino-propyl)-(3-oxo-butyl)-phosphinic acid | C...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260366(CHEMBL4065391)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of human liver cathepsin L peincubated for 5 mins followed by Z-FR-MCA addition by spectrofluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
LigandPNGBDBM50032972(CGP-36216 | (3-Amino-propyl)-ethyl-phosphinic acid...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033024((3-Amino-propyl)-(2-cyclohexyl-ethyl)-phosphinic a...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032996((3-Amino-propyl)-[2-(tetrahydro-pyran-2-yl)-ethyl]...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033008((3-Amino-propyl)-[3-(2-carbamoyl-benzoylamino)-2-h...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260366(CHEMBL4065391)
Affinity DataIC50: 2.02E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 7 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260366(CHEMBL4065391)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human liver cathepsin L peincubated for 5 mins followed by Z-FR-MCA addition by spectrofluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260366(CHEMBL4065391)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human liver cathepsin L peincubated for 5 mins followed by Z-FR-MCA addition by spectrofluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
LigandPNGBDBM50033017((3-Amino-propyl)-cyclohexylmethyl-phosphinic acid ...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032989(CHEMBL113308 | CHEMBL112019 | ((S)-3-Amino-2-hydro...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033014(((R)-3-Amino-2-hydroxy-propyl)-benzyl-phosphinic a...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032989(CHEMBL113308 | CHEMBL112019 | ((S)-3-Amino-2-hydro...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 5.13E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 5.5 uM of substrate Z-FR-MCA measured after 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 5.26E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 6 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 5.72E+3nMAssay Description:Inhibition of cathepsin K (unknown origin) peincubated for 5 mins followed by Z-FR-MCA addition by spectrofluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 5.75E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 8 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
LigandPNGBDBM50032989(CHEMBL113308 | CHEMBL112019 | ((S)-3-Amino-2-hydro...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032987((3-Amino-propyl)-pyridin-2-ylmethyl-phosphinic aci...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032984([3-Amino-2-(4-chloro-phenyl)-2-hydroxy-propyl]-met...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 6.09E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 9 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
LigandPNGBDBM50033004([3-Amino-2-(4-chloro-phenyl)-2-hydroxy-propyl]-but...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 7.17E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 7 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
LigandPNGBDBM50033014(((R)-3-Amino-2-hydroxy-propyl)-benzyl-phosphinic a...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033016((3-Amino-propyl)-(hydroxy-phenyl-methyl)-phosphini...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260367(CHEMBL4102075)
Affinity DataIC50: 8.55E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 7 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
LigandPNGBDBM50033011([3-Amino-2-(4-chloro-phenyl)-propyl]-methyl-phosph...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 9.78E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 5 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
LigandPNGBDBM50033029((3-Amino-propyl)-phenethyl-phosphinic acid | CHEMB...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033018((3-Amino-propyl)-benzyl-phosphinic acid | CHEMBL11...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 1.11E+4nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 4.5 uM of substrate Z-FR-MCA measured after 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 1.15E+4nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 4 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
LigandPNGBDBM50032997(CHEMBL324244 | ((S)-3-Amino-2-hydroxy-propyl)-diet...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260365(CHEMBL4096825)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of cathepsin K (unknown origin) peincubated for 5 mins followed by Z-FR-MCA addition by spectrofluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
LigandPNGBDBM50032995((3-Amino-2-oxo-propyl)-cyclopropylmethyl-phosphini...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032990((3-Amino-propyl)-isobutyl-phosphinic acid | CHEMBL...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033013((3-Amino-propyl)-propyl-phosphinic acid | CHEMBL11...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032997(CHEMBL324244 | ((S)-3-Amino-2-hydroxy-propyl)-diet...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 1.69E+4nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 3.5 uM of substrate Z-FR-MCA measured after 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
LigandPNGBDBM50032994((3-Amino-propyl)-(1-hydroxy-butyl)-phosphinic acid...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033019((3-Amino-propyl)-diisopropoxymethyl-phosphinic aci...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033021((3-Amino-propyl)-dibutoxymethyl-phosphinic acid | ...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033027((3-Amino-propyl)-hexyl-phosphinic acid | CHEMBL113...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033009([3-Amino-2-(4-chloro-phenyl)-propyl]-diethoxymethy...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033012((3-Amino-propyl)-(1,1-difluoro-butyl)-phosphinic a...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033003(CGP-35348 | (3-Amino-propyl)-diethoxymethyl-phosph...)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50032986((3-Amino-propyl)-dipropoxymethyl-phosphinic acid |...)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032985(Bis-(3-amino-propyl)-phosphinic acid | CHEMBL11229...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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