Affinity DataKi: 9.60E+3nMAssay Description:Inhibition of caspase 1 (unknown origin) using N-acetyl-Tyr-Val-Ala-Asp-para-nitroanilide substrate assessed as rate of para-nitroanilide release by ...More data for this Ligand-Target Pair
Affinity DataKi: 1.06E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using N-acetyl-Tyr-Val-Ala-Asp-para-nitroanilide substrate assessed as rate of para-nitroanilide release by ...More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 670nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 7.40E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 4.10E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 22nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 6.50E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 4.00E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 4.80E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 44nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 3.10E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 4.90E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 1.90E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 4.30E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 640nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 360nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 6.30E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 3.30E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Universit£ degli Studi di Torino
Curated by ChEMBL
Universit£ degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 2.00E+4nMAssay Description:Vasodilating activity against phenylephrine-induced contractions in rat thoracic aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 8.20E+3nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 170nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contraction in pres...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Universit£ degli Studi di Torino
Curated by ChEMBL
Universit£ degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 6.30E+3nMAssay Description:Vasodilating activity against phenylephrine-induced contractions in rat thoracic aortaMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Universit£ degli Studi di Torino
Curated by ChEMBL
Universit£ degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Vasodilating activity against phenylephrine-induced contractions in rat thoracic aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contractionMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Universit£ degli Studi di Torino
Curated by ChEMBL
Universit£ degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 860nMAssay Description:Vasodilating activity against phenylephrine-induced contraction in rat thoracic aorta in presence of 1H-[1,2,4]oxadiazolo-[4,3-a]quinoxalin-1-oneMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contraction in pres...More data for this Ligand-Target Pair
Affinity DataEC50: 5.50E+4nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contraction in prese...More data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contraction in pres...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contraction in pres...More data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+3nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contraction in prese...More data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+4nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contraction in prese...More data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+3nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contraction in pres...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Universit£ degli Studi di Torino
Curated by ChEMBL
Universit£ degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 2.00E+4nMAssay Description:Vasodilating activity against phenylephrine-induced contractions in rat thoracic aortaMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Universit£ degli Studi di Torino
Curated by ChEMBL
Universit£ degli Studi di Torino
Curated by ChEMBL
Affinity DataEC50: 1.60E+4nMAssay Description:Vasodilating activity against phenylephrine-induced contraction in rat thoracic aorta in presence of 1H-[1,2,4]oxadiazolo-[4,3-a]quinoxalin-1-oneMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contractionMore data for this Ligand-Target Pair
