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TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50462626(CHEMBL4127893)
Affinity DataKd:  5.26E+3nMAssay Description:Binding affinity to recombinant human N-terminal GSt-tagged TNKS1 (1000 to 1328 residues) expressed in baculovirus infected Sf9 cells by surface plas...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50462627(CHEMBL1958308)
Affinity DataKd:  21nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged TNKS2 (Ser959 to Gly1166 residues) expressed in Escherichia coli by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50462627(CHEMBL1958308)
Affinity DataKd:  520nMAssay Description:Binding affinity to recombinant human N-terminal GSt-tagged TNKS1 (1000 to 1328 residues) expressed in baculovirus infected Sf9 cells by surface plas...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha/beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM11323(CHEMBL177820 | 4,5,6,7-tetrabromo-1H-1,2,3-benzotr...)
Affinity DataKd:  790nMAssay Description:Binding affinity to recombinant human CK2alpha/beta expressed in Escherichia coli by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50188594(CHEMBL1086580 | CHEBI:62878 | US20240279201, Compo...)
Affinity DataKd:  4.20nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged TNKS2 (Ser959 to Gly1166 residues) expressed in Escherichia coli by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50462628(CHEMBL4239155)
Affinity DataKd:  6.5nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged TNKS2 (Ser959 to Gly1166 residues) expressed in Escherichia coli by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50462626(CHEMBL4127893)
Affinity DataKd:  1.25E+3nMAssay Description:Binding affinity to recombinant human PARP1 expressed in baculovirus infected Sf9 cells by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50462629(CHEMBL3594248)
Affinity DataKd:  19nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged TNKS2 (Ser959 to Gly1166 residues) expressed in Escherichia coli by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBcl-2-like protein 1(Human)
Universita Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50480872(CHEMBL582896)
Affinity DataKd:  0.0314nMAssay Description:Binding affinity to Bcl-XL BH3 domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492756(CHEMBL2413566)
Affinity DataKd:  72nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492757(CHEMBL2413581)
Affinity DataKd:  89nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492758(CHEMBL2413580)
Affinity DataKd:  107nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492759(CHEMBL2413569)
Affinity DataKd:  2.80nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492755(CHEMBL2413587)
Affinity DataKd:  84nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492760(CHEMBL2413586)
Affinity DataKd:  191nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492761(CHEMBL2413582)
Affinity DataKd:  201nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492753(CHEMBL2413570)
Affinity DataKd:  3.5nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492762(CHEMBL2413565)
Affinity DataKd:  55nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM227589(Radicicol)
Affinity DataKd:  2.20nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492763(CHEMBL2413573)
Affinity DataKd:  237nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492754(CHEMBL2413568)
Affinity DataKd:  3.60nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492764(CHEMBL2413571)
Affinity DataKd:  10nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50492765(CHEMBL2413579)
Affinity DataKd:  151nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50532223(Hypoestenone)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50532224(CHEMBL4530479)
Affinity DataKd:  21nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50532225(CHEMBL4557055)
Affinity DataKd:  1.74E+3nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50532226(CHEMBL4522895)
Affinity DataKd:  28nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50532227(CHEMBL4447639)
Affinity DataKd:  15nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50532228(CHEMBL4593485)
Affinity DataKd:  217nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50532229(CHEMBL4465174)
Affinity DataKd:  130nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50008057(CHEBI:64153 | BMS-722782 | TANESPIMYCIN)
Affinity DataKd:  388nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50532230(CHEMBL4455666)
Affinity DataKd:  120nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50532231(CHEMBL4584956)
Affinity DataKd:  401nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM227589(Radicicol)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50532232(CHEMBL4570119)
Affinity DataKd:  45nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTubulin beta-3 chain(Human)
Shahid Beheshti University

Curated by ChEMBL
LigandPNGBDBM50424716(Narcotine | Tusscapine | NOSCAPINE)
Affinity DataKd:  579nMAssay Description:Binding affinity to CM5 chip immobilized beta tubulin (unknown origin) assessed as thermodynamic constants by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTubulin beta-3 chain(Human)
Shahid Beheshti University

Curated by ChEMBL
LigandPNGBDBM50546501(CHEMBL4751205)
Affinity DataKd:  133nMAssay Description:Binding affinity to CM5 chip immobilized beta tubulin (unknown origin) assessed as thermodynamic constants by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTubulin beta-3 chain(Human)
Shahid Beheshti University

Curated by ChEMBL
LigandPNGBDBM50546502(CHEMBL4797381)
Affinity DataKd:  22nMAssay Description:Binding affinity to CM5 chip immobilized beta tubulin (unknown origin) assessed as thermodynamic constants by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTubulin beta-3 chain(Human)
Shahid Beheshti University

Curated by ChEMBL
LigandPNGBDBM50546503(CHEMBL4756812)
Affinity DataKd:  37nMAssay Description:Binding affinity to CM5 chip immobilized beta tubulin (unknown origin) assessed as thermodynamic constants by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTubulin beta-3 chain(Human)
Shahid Beheshti University

Curated by ChEMBL
LigandPNGBDBM50546504(CHEMBL4747307)
Affinity DataKd:  374nMAssay Description:Binding affinity to CM5 chip immobilized beta tubulin (unknown origin) assessed as thermodynamic constants by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTubulin beta-3 chain(Human)
Shahid Beheshti University

Curated by ChEMBL
LigandPNGBDBM50546505(CHEMBL4797299)
Affinity DataKd:  132nMAssay Description:Binding affinity to CM5 chip immobilized beta tubulin (unknown origin) assessed as thermodynamic constants by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50570381(CHEMBL4850751)
Affinity DataKd:  18nMAssay Description:Binding affinity to recombinant human HSP90alpha by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50570382(CHEMBL4865803)
Affinity DataKd:  25nMAssay Description:Binding affinity to recombinant human HSP90alpha by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50570383(CHEMBL4854981)
Affinity DataKd:  183nMAssay Description:Binding affinity to recombinant human HSP90alpha by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50570384(CHEMBL4869402)
Affinity DataKd:  25nMAssay Description:Binding affinity to recombinant human HSP90alpha by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50570385(CHEMBL4870060)
Affinity DataKd:  26nMAssay Description:Binding affinity to recombinant human HSP90alpha by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM227589(Radicicol)
Affinity DataKd:  1.80nMAssay Description:Binding affinity to recombinant human HSP90alpha by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(2019-nCoV)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50582092(CHEMBL5091761)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to CM5 sensor chip immobilized SARS-CoV-2 spike glycoprotein assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(2019-nCoV)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50582093(CHEMBL5085757)
Affinity DataKd:  1.91E+4nMAssay Description:Binding affinity to CM5 sensor chip immobilized SARS-CoV-2 spike glycoprotein assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(2019-nCoV)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50582094(CHEMBL5087131)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to CM5 sensor chip immobilized SARS-CoV-2 spike glycoprotein assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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