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TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101257((1R,2S,3R)-1-Benzo[1,3]dioxol-5-yl-3-(2-carboxymet...)
Affinity DataKi:  0.430nMAssay Description:Tested for in vitro inhibition of [125I]-ET-1 binding to CHO cells expressing human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101257((1R,2S,3R)-1-Benzo[1,3]dioxol-5-yl-3-(2-carboxymet...)
Affinity DataKi:  15nMAssay Description:Inhibition of [125I]-ET-1 binding to CHO cells expressing human Endothelin B receptor at a concentration of 1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101268(CHEMBL50232 | [(1R,3R)-1-Benzo[1,3]dioxol-5-yl-3-(...)
Affinity DataIC50:  4.10nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101258(CHEMBL295440 | [(1R,3S)-1-Benzo[1,3]dioxol-5-yl-3-...)
Affinity DataIC50:  5.40nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101271(CHEMBL47868 | [(1R,3S)-1-Benzo[1,3]dioxol-5-yl-3-(...)
Affinity DataIC50:  6.10nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101259(CHEMBL298212 | [(1R,3S)-1-Benzo[1,3]dioxol-5-yl-3-...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101262(3-[2-((1R,3R)-3-Benzo[1,3]dioxol-5-yl-2-carboxymet...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101275(4-[2-((1S,3R)-3-Benzo[1,3]dioxol-5-yl-2-carboxymet...)
Affinity DataIC50:  22nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101261(CHEMBL295140 | {(1R,3S)-1-Benzo[1,3]dioxol-5-yl-5-...)
Affinity DataIC50:  29nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101249(CHEMBL301371 | {2-[(1S,3R)-3-Benzo[1,3]dioxol-5-yl...)
Affinity DataIC50:  31nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101274(CHEMBL430572 | [(1R,3R)-1-Benzo[1,3]dioxol-5-yl-5-...)
Affinity DataIC50:  58nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101254(CHEMBL301723 | [(1R,3R)-1-Benzo[1,3]dioxol-5-yl-5-...)
Affinity DataIC50:  66nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101250(3-[2-((1S,3R)-3-Benzo[1,3]dioxol-5-yl-2-carboxymet...)
Affinity DataIC50:  68nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101247(CHEMBL49850 | [(1R,3S)-1-Benzo[1,3]dioxol-5-yl-5-e...)
Affinity DataIC50:  77nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101251(CHEMBL300000 | [(1R,3S)-1-Benzo[1,3]dioxol-5-yl-3-...)
Affinity DataIC50:  85nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101260(CHEMBL48652 | [(1R,3S)-1-Benzo[1,3]dioxol-5-yl-5-e...)
Affinity DataIC50:  95nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101264(CHEMBL298664 | [(1R,3R)-1-Benzo[1,3]dioxol-5-yl-3-...)
Affinity DataIC50:  96nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101263(CHEMBL49040 | [(1R,3R)-1-Benzo[1,3]dioxol-5-yl-5-e...)
Affinity DataIC50:  96nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101253(CHEMBL417903 | [(1R,3R)-1-Benzo[1,3]dioxol-5-yl-3-...)
Affinity DataIC50:  110nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101269(CHEMBL298922 | [(1R,3R)-1-Benzo[1,3]dioxol-5-yl-3-...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101255(CHEMBL263723 | [(1R,3S)-1-Benzo[1,3]dioxol-5-yl-3-...)
Affinity DataIC50:  310nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101273(CHEMBL48261 | [(1R,3R)-1-Benzo[1,3]dioxol-5-yl-3-(...)
Affinity DataIC50:  330nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101272(CHEMBL299095 | {(1R,3R)-1-Benzo[1,3]dioxol-5-yl-5-...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101267(CHEMBL52110 | [(1R,3S)-1-Benzo[1,3]dioxol-5-yl-5-e...)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288960(CHEMBL156638 | N-[(R)-2-(1H-Indol-3-yl)-1-mercapto...)
Affinity DataIC50:  1.70E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101248(CHEMBL297353 | [(1R,3R)-1-Benzo[1,3]dioxol-5-yl-5-...)
Affinity DataIC50:  3.30E+3nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288958(2-Biphenyl-4-yl-N-((R)-1-mercaptomethyl-2-pyridin-...)
Affinity DataIC50:  5.20E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288964(CHEMBL156740 | Thiophene-2-carboxylic acid [(R)-2-...)
Affinity DataIC50:  5.20E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288957(4-[(R)-2-(1H-Indol-3-yl)-1-mercaptomethyl-ethylcar...)
Affinity DataIC50:  5.40E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288963(2-(4-Benzyloxy-phenyl)-N-[(R)-2-(1H-indol-3-yl)-1-...)
Affinity DataIC50:  6.50E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288961(1-(2-Biphenyl-4-yl-acetyl)-piperidine-4-carboxylic...)
Affinity DataIC50:  6.50E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288962(CHEMBL156964 | N-[(R)-2-(1H-Indol-3-yl)-1-mercapto...)
Affinity DataIC50:  7.70E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288959(CHEMBL421819 | N-((R)-1-Mercaptomethyl-2-phenyl-et...)
Affinity DataIC50:  7.80E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101270(CHEMBL49007 | [(1S,3S)-1-(2-Carboxymethoxy-4-metho...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101252(CHEMBL432499 | [(1R,3R)-1-Benzo[1,3]dioxol-5-yl-3-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101256((1R,3S)-1-Benzo[1,3]dioxol-5-yl-5-ethoxy-2-(1H-tet...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101265(CHEMBL298569 | {(1R,3S)-1-Benzo[1,3]dioxol-5-yl-5-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101266(CHEMBL47563 | [(1S,3R)-1-(2-Carboxymethoxy-4-metho...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to CHO cells expressing recombinant human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed