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TargetOxytocin receptor(Mouse)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataEC50:  62nMAssay Description:Agonist activity at mouse OTR receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077136(CHEMBL3416749)
Affinity DataKd:  61nMAssay Description:Binding affinity to V1aR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397206(CHEMBL2172289)
Affinity DataKd:  1.38nMAssay Description:Binding affinity to SNAP-tagged vasopressin V2 receptor expressed in HEK293 cells after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human V2 receptor expressed in HEK293FT cells incubated for 30 mins by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50326219(CHEMBL1242950 | CHEMBL2206334 | 4-(4-butylpiperidi...)
Affinity DataEC50:  450nMAssay Description:Partial agonist activity at EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells assessed as induction of calci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50139178(CHEMBL3763342)
Affinity DataEC50:  61nMAssay Description:Agonist activity at recombinant human OTR expressed in CHO-DUKX-A2 cells assessed as stimulation of intracellular calcium concentration by calcium 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50401040(CHEMBL2206333)
Affinity DataEC50:  2.51E+4nMAssay Description:Displacement of [3H]NMS from EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells assessed as reduction of [3H]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50139178(CHEMBL3763342)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human V1a receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077134(CHEMBL3416751)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1bR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataEC50:  2.70E+4nMAssay Description:Agonist activity at human V1b receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50077137(CHEMBL3416754)
Affinity DataKd:  1.90nMAssay Description:Binding affinity to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077137(CHEMBL3416754)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1bR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50149891(CHEMBL360055 | 2,2',2''-[1,2,3-BENZENE-TRIYLTRIS(O...)
Affinity DataEC50:  1.74E+5nMAssay Description:Displacement of [3H]NMS from EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells assessed as reduction of [3H]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50459398(CHEMBL4204210)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50077138(CHEMBL3416753)
Affinity DataKon:  0.000182M-1s-1Assay Description:Binding affinity to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells assessed as dissociation constant after 5 to 120 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50326219(CHEMBL1242950 | CHEMBL2206334 | 4-(4-butylpiperidi...)
Affinity DataEC50:  210nMAssay Description:Partial agonist activity at EGFP-fused human full length M1 receptor expressed in HEK293 cells assessed as induction of calcium response by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077139(CHEMBL3416752)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1aR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077136(CHEMBL3416749)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1bR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50139178(CHEMBL3763342)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human OTR expressed in HEK cells assessed as increase in intracellular calcium flux incubated for 45 mins by Indo1-AM dye based f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50326219(CHEMBL1242950 | CHEMBL2206334 | 4-(4-butylpiperidi...)
Affinity DataEC50:  740nMAssay Description:Partial agonist activity at human full length M1 receptor expressed in HEK293 cells assessed as induction of calcium response by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50459398(CHEMBL4204210)
Affinity DataEC50:  62nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293FT cells incubated for 30 mins by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataEC50:  250nMAssay Description:Agonist activity at EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells assessed as induction of calcium respo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293FT cells incubated for 30 mins by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataEC50:  1.50E+4nMAssay Description:Agonist activity at human M3 receptor in HEK293 cells assessed as induction of calcium response by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50326219(CHEMBL1242950 | CHEMBL2206334 | 4-(4-butylpiperidi...)
Affinity DataEC50:  720nMAssay Description:Partial agonist activity at EGFP-fused human M1 receptor N-terminal truncated at 11 residues expressed in HEK293 cells assessed as induction of calci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human OTR receptor expressed in CHO cells co-expressing NFAT-luciferase incubated for 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077137(CHEMBL3416754)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1aR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50177593((5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)...)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at V2 receptor (unknown origin) by cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50459404(CHEMBL4205046)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human V2 receptor expressed in human HeLa cells assessed as cAMP accumulation incubated for 10 mins by radioimmunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  810nMAssay Description:Agonist activity at human V2 receptor expressed in HEK293FT cells incubated for 30 mins by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50077135(CHEMBL3416750)
Affinity DataKd:  1.40nMAssay Description:Binding affinity to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077138(CHEMBL3416753)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1bR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human V2 receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human V1b receptor expressed in HEK293FT cells incubated for 30 mins by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50459390(CHEMBL4216174)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human OTR expressed in HEK cells assessed as increase in intracellular calcium flux incubated for 45 mins by Indo1-AM dye based f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50077139(CHEMBL3416752)
Affinity DataKd:  2.10nMAssay Description:Binding affinity to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetOxytocin receptor(Mouse)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50459398(CHEMBL4204210)
Affinity DataEC50:  18nMAssay Description:Agonist activity at mouse OTR receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  8nMAssay Description:Agonist activity at SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells assessed as intracellular calcium flux after 3 mins by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077134(CHEMBL3416751)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V2R (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50077138(CHEMBL3416753)
Affinity DataKd:  1.60nMAssay Description:Binding affinity to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077137(CHEMBL3416754)
Affinity DataKd:  353nMAssay Description:Binding affinity to V2R (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077139(CHEMBL3416752)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V2R (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetStromal cell-derived factor 1(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369279(CHEMBL4166454)
Affinity DataKd:  780nMAssay Description:Binding affinity to CXCL12 (unknown origin) assessed as changes in tryptophan fluorescence intensityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50077134(CHEMBL3416751)
Affinity DataKon:  0.000315M-1s-1Assay Description:Binding affinity to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells assessed as dissociation constant after 5 to 120 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397209(CHEMBL2172291)
Affinity DataKd:  2.53nMAssay Description:Binding affinity to SNAP-tagged vasopressin V2 receptor expressed in HEK293 cells after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077135(CHEMBL3416750)
Affinity DataKd:  20nMAssay Description:Binding affinity to V1aR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077135(CHEMBL3416750)
Affinity DataKd:  31nMAssay Description:Binding affinity to V2R (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077138(CHEMBL3416753)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1aR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
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