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TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50494549(CHEMBL3093327)
Affinity DataKi:  0.124nMAssay Description:Binding affinity to rat adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268151(1-Ethyl-8-(4-(4-(4-trifluoromethylbenzyl)piperazin...)
Affinity DataKi:  0.157nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268107(CHEMBL485862 | CHEMBL500634 | N-(2-(2-phenyl-6-(4-...)
Affinity DataKd:  0.170nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268109(8-(4-(4-(4-chlorobenzyl)piperazin-1-ylsulfonyl)phe...)
Affinity DataKi:  0.215nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268164(1-Ethyl-8-(4-(4-(3-trifluoromethylbenzyl)piperazin...)
Affinity DataKi:  0.281nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268163(1-Propyl-8-(4-(4-(4-trifluoromethylbenzyl)piperazi...)
Affinity DataKi:  0.303nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Mouse)
Institute

Curated by ChEMBL
LigandPNGBDBM50268232(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKd:  0.351nMAssay Description:Displacement of [3H]PSB-603 from mouse recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268129(8-(4-(4-(4-chlorobenzyl)piperazin-1-ylsulfonyl)phe...)
Affinity DataKi:  0.393nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268232(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKd:  0.403nMAssay Description:Binding affinity to human recombinant adenosine A2B receptor expressed in CHO cells by saturation experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268231(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.406nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268107(CHEMBL485862 | CHEMBL500634 | N-(2-(2-phenyl-6-(4-...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268150(8-(4-(4-(3-Fluorobenzyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.446nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268233(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.473nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268232(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.553nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268132(8-(4-(4-(4-Fluorobenzyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.595nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268130(8-(4-(4-(3-Chlorobenzyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268232(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKd:  0.652nMAssay Description:Binding affinity to human recombinant adenosine A2B receptor expressed in CHO cells by kinetic experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268149(1-Ethyl-8-(4-(4-(3-fluorobenzyl)piperazine-1-sulfo...)
Affinity DataKi:  0.695nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50494549(CHEMBL3093327)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268165(1-Propyl-8-(4-(4-(3-trifluoromethylbenzyl)piperazi...)
Affinity DataKi:  0.775nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268110(8-(4-(4-(3-Chlorobenzyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.782nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268181(8-(4-(4-(4-Methylbenzyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.858nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268210(8-(4-(4-Benzo[1,3]dioxol-5-ylmethylpiperazine-1-su...)
Affinity DataKi:  0.875nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268209(8-(4-(4-(4-Methoxybenzyl)piperazine-1-sulfonyl)phe...)
Affinity DataKi:  0.944nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268211(8-(4-(4-Benzo[1,3]dioxol-5-ylmethylpiperazine-1-su...)
Affinity DataKi:  1.06nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268232(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataIC50: 1.13nMAssay Description:Antagonist activity at adenosine A2B receptor in human Jurkat T cells assessed as inhibition of NECA-induced increase in intracellular calcium concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50086170(CHEMBL1628266 | N-(4-Cyano-phenyl)-2-[4-(2,6-dioxo...)
Affinity DataKd:  1.13nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268108(8-(4-(4-benzylpiperazin-1-ylsulfonyl)phenyl)-1-eth...)
Affinity DataKi:  1.15nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268182(1-Ethyl-8-(4-(4-(4-methoxybenzyl)piperazine-1-sulf...)
Affinity DataKi:  1.19nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268085(CHEMBL490262 | SB-298 | CHEMBL521280 | N-(2-hydrox...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268131(1-Ethyl-8-(4-(4-(4-fluorobenzyl)piperazine-1-sulfo...)
Affinity DataKi:  1.27nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50190709(8-[4-(4-benzylpiperazide-1-sulfonyl)phenyl]-1-prop...)
Affinity DataKi:  1.33nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268180(1-Ethyl-8-(4-(4-(4-methylbenzyl)piperazine-1-sulfo...)
Affinity DataKi:  1.58nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268163(1-Propyl-8-(4-(4-(4-trifluoromethylbenzyl)piperazi...)
Affinity DataIC50: 1.62nMAssay Description:Antagonist activity at adenosine A2B receptor in human Jurkat T cells assessed as inhibition of NECA-induced increase in intracellular calcium concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50229885(N-(benzo[d][1,3]dioxol-5-yl)-2-(5-(2,6-dioxo-1,3-d...)
Affinity DataKd:  1.65nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268110(8-(4-(4-(3-Chlorobenzyl)piperazine-1-sulfonyl)phen...)
Affinity DataIC50: 1.91nMAssay Description:Antagonist activity at adenosine A2B receptor in human Jurkat T cells assessed as inhibition of NECA-induced increase in intracellular calcium concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50086170(CHEMBL1628266 | N-(4-Cyano-phenyl)-2-[4-(2,6-dioxo...)
Affinity DataKi:  1.97nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268245(8-(4-(4-(4-Methoxyphenyl)piperazine-1-sulfonyl)phe...)
Affinity DataKi:  1.99nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268164(1-Ethyl-8-(4-(4-(3-trifluoromethylbenzyl)piperazin...)
Affinity DataIC50: 2.29nMAssay Description:Antagonist activity at adenosine A2B receptor in human Jurkat T cells assessed as inhibition of NECA-induced increase in intracellular calcium concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268257(N-(1-Benzylpiperidin-4-yl)-4-(2,6-dioxo-1-propyl-2...)
Affinity DataKi:  3.03nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268150(8-(4-(4-(3-Fluorobenzyl)piperazine-1-sulfonyl)phen...)
Affinity DataIC50: 3.23nMAssay Description:Antagonist activity at adenosine A2B receptor in human Jurkat T cells assessed as inhibition of NECA-induced increase in intracellular calcium concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Mouse)
Institute

Curated by ChEMBL
LigandPNGBDBM50086170(CHEMBL1628266 | N-(4-Cyano-phenyl)-2-[4-(2,6-dioxo...)
Affinity DataKi:  3.39nMAssay Description:Binding affinity to mouse adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268165(1-Propyl-8-(4-(4-(3-trifluoromethylbenzyl)piperazi...)
Affinity DataIC50: 3.56nMAssay Description:Antagonist activity at adenosine A2B receptor in human Jurkat T cells assessed as inhibition of NECA-induced increase in intracellular calcium concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50190709(8-[4-(4-benzylpiperazide-1-sulfonyl)phenyl]-1-prop...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268129(8-(4-(4-(4-chlorobenzyl)piperazin-1-ylsulfonyl)phe...)
Affinity DataIC50: 3.64nMAssay Description:Antagonist activity at adenosine A2B receptor in human Jurkat T cells assessed as inhibition of NECA-induced increase in intracellular calcium concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268108(8-(4-(4-benzylpiperazin-1-ylsulfonyl)phenyl)-1-eth...)
Affinity DataIC50: 4.49nMAssay Description:Antagonist activity at adenosine A2B receptor in human Jurkat T cells assessed as inhibition of NECA-induced increase in intracellular calcium concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268182(1-Ethyl-8-(4-(4-(4-methoxybenzyl)piperazine-1-sulf...)
Affinity DataIC50: 5.26nMAssay Description:Antagonist activity at adenosine A2B receptor in human Jurkat T cells assessed as inhibition of NECA-induced increase in intracellular calcium concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50268210(8-(4-(4-Benzo[1,3]dioxol-5-ylmethylpiperazine-1-su...)
Affinity DataIC50: 5.34nMAssay Description:Antagonist activity at adenosine A2B receptor in human Jurkat T cells assessed as inhibition of NECA-induced increase in intracellular calcium concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50084860(3-(3-Hydroxy-propyl)-8-[2-(3-methoxy-phenyl)-vinyl...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]MSX-2 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
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