Compile Data Set for Download or QSAR
Found 13 with Last Name = 'cairati' and Initial = 's'
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM50240586(CHEMBL4098982)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM50240587(CHEMBL4070316)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM32609(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 36b)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM50240589(CHEMBL4091245)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM50240592(CHEMBL4097534)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM50240588(CHEMBL4079500)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM50240586(CHEMBL4098982)
Affinity DataIC50:  91nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM50535120(CHEMBL4451097)
Affinity DataIC50:  370nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM50535123(CHEMBL4552544)
Affinity DataIC50:  1.09E+3nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM50535122(CHEMBL4452878)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM50535121(CHEMBL4452014)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM50535119(CHEMBL4457255)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)

Curated by ChEMBL
LigandPNGBDBM36363(CID6851947 | PAC-1 | US10166229, Example PAC-1)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed