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TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.110nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.120nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.130nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.160nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKi:  0.180nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50166224(CHEMBL410567 | Vasopressin Analogue)
Affinity DataKi:  0.180nMAssay Description:Binding affinity against rat vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.200nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.240nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50103475(Pmp-Tyr-Ile-Thr-Asn-Cys-Pro-Orn-phe(I,N3)-NH2 | Pm...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.310nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.310nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKi:  0.460nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.470nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50103477(CHEMBL386180 | Pmp-Tyr-Ile-Thr-Asn-Cys-Pro-Orn-phe...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.650nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50166219(CHEMBL264101 | Vasopressin Analogue)
Affinity DataKi:  0.800nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  1.40nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  1.60nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50103478(CHEMBL406670 | Pmp-Tyr(Me)-Ile-Thr-Asn-Cys-Pro-Orn...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50166225(CHEMBL410401 | Vasopressin Analogue)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKi:  3nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  4.80nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  8nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  10nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038605(3-N3-C6H4CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-...)
Affinity DataKi:  17.8nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50166223(CHEMBL265137 | Vasopressin Analogue)
Affinity DataKi:  18nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKi:  18nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50103476(CHEMBL412559 | Pmp-Tyr-Ile-Thr-Asn-Cys-Pro-Orn-phe...)
Affinity DataKi:  18nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50166218((2S)-2-[(2S)-2-[(2R)-2-azaniumyl-3-(4-benzoylpheny...)
Affinity DataKi:  20nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038600(4-N3-C6H4CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-...)
Affinity DataKi:  20nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50166222(CHEMBL410673 | Vasopressin Analogue)
Affinity DataKi:  24nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  37.7nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50166227(CHEMBL439430 | Vasopressin Analogue)
Affinity DataKi:  115nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50166220((2S)-2-[(2S)-2-[(2S)-2-azaniumyl-3-(4-benzoylpheny...)
Affinity DataKi:  148nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50166226((2S)-2-[(2S)-2-[(2R)-2-[2-azaniumyl-3-(4-benzoylph...)
Affinity DataKi:  462nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50166221(CHEMBL408657 | Vasopressin Analogue)
Affinity DataKi:  1.49E+3nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  1.60E+4nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50103475(Pmp-Tyr-Ile-Thr-Asn-Cys-Pro-Orn-phe(I,N3)-NH2 | Pm...)
Affinity DataIC50:  0.320nMAssay Description:Ability to inhibit OT-induced inositol phosphate accumulation was determined in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50103475(Pmp-Tyr-Ile-Thr-Asn-Cys-Pro-Orn-phe(I,N3)-NH2 | Pm...)
Affinity DataKd:  0.25nMAssay Description:Dissociation constant value of the compound was determined for human OT-receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKd:  0.0540nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKd:  0.0400nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50103475(Pmp-Tyr-Ile-Thr-Asn-Cys-Pro-Orn-phe(I,N3)-NH2 | Pm...)
Affinity DataKd:  0.25nMAssay Description:Dissociation constant value of the compound was determined for human OT-receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKd:  0.190nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKd:  0.150nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed