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Report error Found 2813 with Last Name = 'casimiro-garcia' and Initial = 'a'
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50: >1.20E+4nMpH: 7.2 T: 2°CAssay Description:Human PPAR alpha receptor was expressed as recombinant glutathione-S-transferase (GST)-fusion proteins in Escherichia coli. The purified GST-hPPAR al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2009
Entry Details Article
PubMed
LigandPNGBDBM33286(racemic | phenylpropanoic acid derivative, 17b)
Affinity DataEC50:  5.70E+3nMpH: 7.2 T: 2°CAssay Description:Human PPAR alpha receptor was expressed as recombinant glutathione-S-transferase (GST)-fusion proteins in Escherichia coli. The purified GST-hPPAR al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2009
Entry Details Article
PubMed
LigandPNGBDBM33287(racemic | phenylpropanoic acid derivative, 17c)
Affinity DataEC50:  8.50E+3nMpH: 7.2 T: 2°CAssay Description:Human PPAR alpha receptor was expressed as recombinant glutathione-S-transferase (GST)-fusion proteins in Escherichia coli. The purified GST-hPPAR al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2009
Entry Details Article
PubMed
LigandPNGBDBM33290(phenylpropanoic acid derivative, 17f)
Affinity DataEC50: >2.00E+4nMpH: 7.2 T: 2°CAssay Description:Human PPAR alpha receptor was expressed as recombinant glutathione-S-transferase (GST)-fusion proteins in Escherichia coli. The purified GST-hPPAR al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2009
Entry Details Article
PubMed
LigandPNGBDBM33291(racemic | phenylpropanoic acid derivative, 17g)
Affinity DataEC50: >1.00E+5nMpH: 7.2 T: 2°CAssay Description:Human PPAR alpha receptor was expressed as recombinant glutathione-S-transferase (GST)-fusion proteins in Escherichia coli. The purified GST-hPPAR al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2009
Entry Details Article
PubMed
LigandPNGBDBM33292(racemic | phenylpropanoic acid derivative, 17h)
Affinity DataEC50: >1.00E+5nMpH: 7.2 T: 2°CAssay Description:Human PPAR alpha receptor was expressed as recombinant glutathione-S-transferase (GST)-fusion proteins in Escherichia coli. The purified GST-hPPAR al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2009
Entry Details Article
PubMed
TargetPantetheinase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM480973(US10906888, Example 190)
Affinity DataKd:  20nMAssay Description:Binding affinity to recombinant N-terminal FLAG/His6-tagged human vanin-1 expressed in CHO cells assessed as dissociation constant by surface plasmon...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetPantetheinase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM480978(US10906888, Example 196 | US10906888, Example 197 ...)
Affinity DataKd:  7.20nMAssay Description:Binding affinity to recombinant N-terminal FLAG/His6-tagged human vanin-1 expressed in CHO cells assessed as dissociation constant by surface plasmon...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetPantetheinase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM480981(US10906888, Example 200 | US10906888, Example 199 ...)
Affinity DataKd:  37nMAssay Description:Binding affinity to recombinant N-terminal FLAG/His6-tagged human vanin-1 expressed in CHO cells assessed as dissociation constant by surface plasmon...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetGlucose-induced degradation protein 4 homolog(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50589800(CHEMBL5197897)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity to recombinant GID4 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetGlucose-induced degradation protein 4 homolog(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50621188(CHEMBL5426366)
Affinity DataKd:  1.50E+4nMAssay Description:Binding affinity to recombinant GID4 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetGlucose-induced degradation protein 4 homolog(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50621189(CHEMBL5414824)
Affinity DataKd:  9.00E+3nMAssay Description:Binding affinity to recombinant GID4 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetGlucose-induced degradation protein 4 homolog(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50621190(CHEMBL5405098)
Affinity DataKd:  3.40E+3nMAssay Description:Binding affinity to recombinant GID4 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPDBSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlucose-induced degradation protein 4 homolog(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50621191(CHEMBL5435433)
Affinity DataKd:  2.70E+3nMAssay Description:Binding affinity to recombinant GID4 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetGlucose-induced degradation protein 4 homolog(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50621192(CHEMBL5411414)
Affinity DataKd:  2.40E+4nMAssay Description:Binding affinity to recombinant GID4 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetGlucose-induced degradation protein 4 homolog(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50621193(CHEMBL5411984)
Affinity DataKd:  500nMAssay Description:Binding affinity to recombinant GID4 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetGlucose-induced degradation protein 4 homolog(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50621194(CHEMBL5393907)
Affinity DataKd:  300nMAssay Description:Binding affinity to recombinant GID4 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetGlucose-induced degradation protein 4 homolog(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50589806(CHEMBL5177469)
Affinity DataKd:  81nMAssay Description:Binding affinity to recombinant GID4 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50347564(CHEMBL1801741)
Affinity DataEC50:  89nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347565(CHEMBL1801743)
Affinity DataEC50:  90nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347574(CHEMBL1801742)
Affinity DataEC50:  165nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347570(CHEMBL1801744)
Affinity DataEC50:  175nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347563(CHEMBL1801740)
Affinity DataEC50:  212nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347573(CHEMBL1801739)
Affinity DataEC50:  264nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347569(CHEMBL1801734)
Affinity DataEC50:  295nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347566(CHEMBL1801738)
Affinity DataEC50:  494nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50282484(2-Ethyl-5,7-dimethyl-3-{5-[2-(1H-tetrazol-5-yl)-ph...)
Affinity DataEC50:  574nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347567(CHEMBL1801712)
Affinity DataEC50:  591nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347568(CHEMBL1801735)
Affinity DataEC50:  762nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50049240((+-)-5-((4-(2-(5-ethyl-2-pyridinyl)ethoxy)phenyl)m...)
Affinity DataEC50:  1.28E+3nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347571(CHEMBL1801714)
Affinity DataEC50:  1.32E+3nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347572(CHEMBL1801737)
Affinity DataEC50:  1.34E+3nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50043280(4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimi...)
Affinity DataEC50:  1.52E+3nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50282478(2-Butyl-5,7-dimethyl-3-{5-[2-(1H-tetrazol-5-yl)-ph...)
Affinity DataEC50:  2.20E+3nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347576(CHEMBL1801713)
Affinity DataEC50:  2.62E+3nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50009718(CHEMBL7550 | 2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetraz...)
Affinity DataEC50: >2.00E+4nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50347575(CHEMBL1801736)
Affinity DataEC50:  1.82E+3nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50426774(CHEMBL2322437)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at PPARbeta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426774(CHEMBL2322437)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at PPARalpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426776(CHEMBL2322176)
Affinity DataEC50:  295nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426777(CHEMBL2322175)
Affinity DataEC50:  42nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426778(CHEMBL2322174)
Affinity DataEC50:  4.47E+3nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426779(CHEMBL2322173)
Affinity DataEC50: >2.50E+4nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426780(CHEMBL2322172)
Affinity DataEC50:  3.64E+3nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426781(CHEMBL2322451)
Affinity DataEC50:  3.58E+3nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426782(CHEMBL2322450)
Affinity DataEC50:  449nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426783(CHEMBL2322449)
Affinity DataEC50:  108nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426784(CHEMBL2322448)
Affinity DataEC50:  159nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426785(CHEMBL2322447)
Affinity DataEC50:  20nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50426786(CHEMBL2322446)
Affinity DataEC50:  187nMAssay Description:Partial agonist activity at human PPARgamma-LBD/Gal4 DNA binding domain by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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