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TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345484(N4-Benzyloxycytidine-5'-triphosphate | CHEMBL17848...)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50241299({[(2R,3S,4R,5R)-5-(2,4-dioxo-1,2,3,4-tetrahydropyr...)
Affinity DataEC50:  1.31E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345491(Uridine-5'-allose-1'-tetraphosphate | CHEMBL178488...)
Affinity DataEC50:  770nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118239(uridine 5'-(trihydrogen diphosphate) | UDP | Uridi...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50205405(({[({[(2R,3S,4R,5R)-4-amino-5-(2,4-dioxo-1,2,3,4-t...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50270551(P1,P4-di(uridine 5'-)beta,gamma-difluoromethylenet...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345494(P1-(Uridine-5'-)P4-(2'-deoxy-2'-acetamidoglucose-1...)
Affinity DataEC50:  5.46E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271292(Uridine-5'-alpha-glycerol-tetraphosphate | CHEMBL4...)
Affinity DataEC50:  8.19E+3nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50270545(Uridine-5'-glucose-1'-tetraphosphate | CHEMBL49913...)
Affinity DataEC50:  7.83E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50270542(Uridine-5'-cyclohexane-tetraphosphate | CHEMBL4748...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50270546(Uridine-5'-galactose-1'-tetraphosphate | CHEMBL444...)
Affinity DataEC50:  4.85E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271222(({[({[(2R,3S,4R,5R)-4-(carbamoylamino)-5-(2,4-diox...)
Affinity DataEC50:  4.64E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271187([dichloro({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-(4-ox...)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human P2Y2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271289(Uridine-5'-methyl-tetraphosphate | CHEMBL519991)
Affinity DataEC50:  4.00E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50270546(Uridine-5'-galactose-1'-tetraphosphate | CHEMBL444...)
Affinity DataEC50:  1.77E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345483(N4-t-Butyloxycytidine-5'-triphosphate | CHEMBL1784...)
Affinity DataEC50:  2.11E+3nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50205413(P(1),P(4)-bis(uridin-5'-yl) tetraphosphate | P1,P4...)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345486(N4-Phenylpropoxycytidine-5'-triphosphate | CHEMBL1...)
Affinity DataEC50:  640nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50241299({[(2R,3S,4R,5R)-5-(2,4-dioxo-1,2,3,4-tetrahydropyr...)
Affinity DataEC50:  870nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50270554(P1-(2-thiouridine 5'-)-P4-(2'-deoxycytidine 5'-)te...)
Affinity DataEC50:  1.05E+3nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345492(Uridine-5'-mannose-1'-tetraphosphate | CHEMBL17848...)
Affinity DataEC50:  4.48E+3nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345495(P1-(Uridine-5'-)P4-(glucuronic acid-1'-)tetraphosp...)
Affinity DataEC50:  227nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50270546(Uridine-5'-galactose-1'-tetraphosphate | CHEMBL444...)
Affinity DataEC50:  8.19E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271292(Uridine-5'-alpha-glycerol-tetraphosphate | CHEMBL4...)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50270555({[(2R,3S,5R)-5-(2-amino-6-oxo-6,9-dihydro-3H-purin...)
Affinity DataEC50:  540nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271253(4-Thio-uridine-5'-tetraphosphate | CHEMBL521451)
Affinity DataEC50:  280nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271291(Uridine-5'-(2-cyanoethyl)-tetraphosphate | CHEMBL4...)
Affinity DataEC50:  1.96E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271253(4-Thio-uridine-5'-tetraphosphate | CHEMBL521451)
Affinity DataEC50:  6.46E+3nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50270549(P1-((2-benzyl-1,3-dioxolo-4-yl)uridine 5')P3-(5-io...)
Affinity DataEC50:  9.97E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345486(N4-Phenylpropoxycytidine-5'-triphosphate | CHEMBL1...)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50270547(Uridine-5'-mannose-6'-tetraphosphate | CHEMBL50812...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50270545(Uridine-5'-glucose-1'-tetraphosphate | CHEMBL49913...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345491(Uridine-5'-allose-1'-tetraphosphate | CHEMBL178488...)
Affinity DataEC50:  183nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345482(N4-Ethoxycytidine-5'-triphosphate | CHEMBL1784890)
Affinity DataEC50:  877nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345485(N4-Phenylethoxycytidine-5'-triphosphate | CHEMBL17...)
Affinity DataEC50:  1.21E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50241299({[(2R,3S,4R,5R)-5-(2,4-dioxo-1,2,3,4-tetrahydropyr...)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345496(P1-(Uridine-5'-)P4-(3'-deoxy-3'-fluoroglucose-1'-)...)
Affinity DataEC50:  950nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271290(Uridine-5'-methyl(C-P)-tetraphosphate | CHEMBL4839...)
Affinity DataEC50:  4.18E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271101([(2R,3S,4R,5R)-5-(5-amino-2,4-dioxo-3,4-dihydropyr...)
Affinity DataEC50:  610nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271289(Uridine-5'-methyl-tetraphosphate | CHEMBL519991)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345497(P1-(N4-Benzyloxycytidine-5'-)P4-(3'-deoxy-3'-fluor...)
Affinity DataEC50:  7.51E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271223(({[({[(2R,3S,4S,5R)-3,4-dihydroxy-5-(4-oxo-2-sulfa...)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50271222(({[({[(2R,3S,4R,5R)-4-(carbamoylamino)-5-(2,4-diox...)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345495(P1-(Uridine-5'-)P4-(glucuronic acid-1'-)tetraphosp...)
Affinity DataEC50:  490nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50345498(P1-(N4-Methoxycytidine-5'-)P4-(3'-deoxy-3'-fluorog...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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