Compile Data Set for Download or QSAR
Found 173 with Last Name = 'cena' and Initial = 'c'
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50018796(2,6-Dimethyl-4-(3-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072809(4-[2-(4-Cyano-furazan-3-ylmethoxy)-phenyl]-2,6-dim...)
Affinity DataKi:  4.70nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072811(2,6-Dimethyl-4-[2-(4-methyl-5-oxy-furazan-3-ylmeth...)
Affinity DataKi:  18nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072818(4-[2-(4-Cyano-5-oxy-furazan-3-ylmethoxy)-phenyl]-2...)
Affinity DataKi:  21nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072803(2,6-Dimethyl-4-[2-(4-methyl-furazan-3-ylmethoxy)-p...)
Affinity DataKi:  27nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072814(4-[2-(4-Cyano-2-oxy-furazan-3-ylmethoxy)-phenyl]-2...)
Affinity DataKi:  30nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072810(2,6-Dimethyl-4-[2-(4-methyl-2-oxy-furazan-3-ylmeth...)
Affinity DataKi:  32nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072816(2,6-Dimethyl-4-[2-(2-nitrooxy-ethoxy)-phenyl]-1,4-...)
Affinity DataKi:  38nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072804(4-[3-(4-Cyano-2-oxy-furazan-3-ylmethoxy)-phenyl]-2...)
Affinity DataKi:  220nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072817(4-[3-(4-Cyano-5-oxy-furazan-3-ylmethoxy)-phenyl]-2...)
Affinity DataKi:  230nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072806(4-[3-(4-Cyano-furazan-3-ylmethoxy)-phenyl]-2,6-dim...)
Affinity DataKi:  270nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072813(2,6-Dimethyl-4-[3-(4-methyl-2-oxy-furazan-3-ylmeth...)
Affinity DataKi:  280nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072812(2,6-Dimethyl-4-[3-(4-methyl-furazan-3-ylmethoxy)-p...)
Affinity DataKi:  320nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072807(4-[2-(4-Carbamoyl-2-oxy-furazan-3-ylmethoxy)-pheny...)
Affinity DataKi:  350nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072800(2,6-Dimethyl-4-[3-(4-methyl-5-oxy-furazan-3-ylmeth...)
Affinity DataKi:  370nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072801(4-[2-(4-Carbamoyl-furazan-3-ylmethoxy)-phenyl]-2,6...)
Affinity DataKi:  400nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072802(2,6-Dimethyl-4-[3-(2-nitrooxy-ethoxy)-phenyl]-1,4-...)
Affinity DataKi:  440nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072815(4-[2-(4-Carbamoyl-5-oxy-furazan-3-ylmethoxy)-pheny...)
Affinity DataKi:  670nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072808(4-[3-(4-Carbamoyl-5-oxy-furazan-3-ylmethoxy)-pheny...)
Affinity DataKi:  920nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072819(4-[3-(4-Carbamoyl-2-oxy-furazan-3-ylmethoxy)-pheny...)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072805(4-[3-(4-Carbamoyl-furazan-3-ylmethoxy)-phenyl]-2,6...)
Affinity DataKi:  2.30E+3nMAssay Description:Binding affinity for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50018796(2,6-Dimethyl-4-(3-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  2.60nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataIC50:  2.70nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072809(4-[2-(4-Cyano-furazan-3-ylmethoxy)-phenyl]-2,6-dim...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072818(4-[2-(4-Cyano-5-oxy-furazan-3-ylmethoxy)-phenyl]-2...)
Affinity DataIC50:  27nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072811(2,6-Dimethyl-4-[2-(4-methyl-5-oxy-furazan-3-ylmeth...)
Affinity DataIC50:  40nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072803(2,6-Dimethyl-4-[2-(4-methyl-furazan-3-ylmethoxy)-p...)
Affinity DataIC50:  59nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072814(4-[2-(4-Cyano-2-oxy-furazan-3-ylmethoxy)-phenyl]-2...)
Affinity DataIC50:  67nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072810(2,6-Dimethyl-4-[2-(4-methyl-2-oxy-furazan-3-ylmeth...)
Affinity DataIC50:  72nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072816(2,6-Dimethyl-4-[2-(2-nitrooxy-ethoxy)-phenyl]-1,4-...)
Affinity DataIC50:  85nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Università degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50131622(4-Chloro-5-(3-fluoro-4-methoxy-phenyl)-1-(4-methan...)
Affinity DataIC50:  90nMAssay Description:Activity of COX2 in human heparinized blood assessed as inhibition of LPS-induced PGE2 production after 24 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Università degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50131593(4-[4-Chloro-5-(3-fluoro-4-methoxy-phenyl)-imidazol...)
Affinity DataIC50:  100nMAssay Description:Activity of COX2 in human heparinized blood assessed as inhibition of LPS-induced PGE2 production after 24 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University of Torino

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  100nMAssay Description:Antagonistic activity against TP-receptor by inhibition of U 46619-induced contraction of isolated guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University of Torino

Curated by ChEMBL
LigandPNGBDBM50277998(CHEMBL4174786)
Affinity DataIC50:  310nMAssay Description:Inhibition of AKR1C3 (unknown origin) using S-tetralol as substrate in presence of NADP+ by fluorimteryMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University of Torino

Curated by ChEMBL
LigandPNGBDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataIC50:  440nMAssay Description:Inhibition of type-1 human steroid 5-alpha-reductaseMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University of Torino

Curated by ChEMBL
LigandPNGBDBM50278013(CHEMBL4166887)
Affinity DataIC50:  480nMAssay Description:Thromboxane (TXA2) receptor antagonist activity using human plateletMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072817(4-[3-(4-Cyano-5-oxy-furazan-3-ylmethoxy)-phenyl]-2...)
Affinity DataIC50:  500nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072804(4-[3-(4-Cyano-2-oxy-furazan-3-ylmethoxy)-phenyl]-2...)
Affinity DataIC50:  500nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C2(Homo sapiens (Human))
University of Torino

Curated by ChEMBL
LigandPNGBDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataIC50:  530nMAssay Description:Antagonistic activity against TP-receptor by inhibition of U 46619-induced contraction of isolated guinea pig tracheaMore data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit 2(Homo sapiens (Human))
University of Torino

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  540nMAssay Description:Thromboxane (TXA2) receptor antagonist activity using human plateletMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072806(4-[3-(4-Cyano-furazan-3-ylmethoxy)-phenyl]-2,6-dim...)
Affinity DataIC50:  590nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome c oxidase subunit 2(Homo sapiens (Human))
University of Torino

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  610nMAssay Description:Antagonistic activity against TP-receptor by inhibition of U 46619-induced contraction of isolated guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072813(2,6-Dimethyl-4-[3-(4-methyl-2-oxy-furazan-3-ylmeth...)
Affinity DataIC50:  610nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072812(2,6-Dimethyl-4-[3-(4-methyl-furazan-3-ylmethoxy)-p...)
Affinity DataIC50:  720nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072807(4-[2-(4-Carbamoyl-2-oxy-furazan-3-ylmethoxy)-pheny...)
Affinity DataIC50:  780nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072800(2,6-Dimethyl-4-[3-(4-methyl-5-oxy-furazan-3-ylmeth...)
Affinity DataIC50:  820nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072801(4-[2-(4-Carbamoyl-furazan-3-ylmethoxy)-phenyl]-2,6...)
Affinity DataIC50:  880nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM50072802(2,6-Dimethyl-4-[3-(2-nitrooxy-ethoxy)-phenyl]-1,4-...)
Affinity DataIC50:  970nMAssay Description:Inhibitory concentration for L-type [Ca2+] channels was measured through displacement of [3H]nitrendipine on rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Università degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  1.30E+3nMAssay Description:Activity of COX2 in human heparinized blood assessed as inhibition of LPS-induced PGE2 production after 24 hrsMore data for this Ligand-Target Pair
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