Compile Data Set for Download or QSAR
Report error Found 159 with Last Name = 'chebib' and Initial = 'm'
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50481220(CHEMBL608389)
Affinity DataEC50:  1.37E+4nMAssay Description:Modulatory activity at human GABAA alpha-1-beta-2-gamma-2L receptor expressed in Xenopus laevis oocytes assessed as potentiation of of GABA EC5-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50481221(CHEMBL595673)
Affinity DataEC50:  1.50E+4nMAssay Description:Modulatory activity at human GABAA alpha-1-beta-2-gamma-2L receptor expressed in Xenopus laevis oocytes assessed as potentiation of of GABA EC5-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50481222(CHEMBL595422)
Affinity DataEC50:  1.22E+4nMAssay Description:Modulatory activity at human GABAA alpha-1-beta-2-gamma-2L receptor expressed in Xenopus laevis oocytes assessed as potentiation of of GABA EC5-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50481223(CHEMBL609751)
Affinity DataEC50:  6.68E+3nMAssay Description:Modulatory activity at human GABAA alpha-1-beta-2-gamma-2L receptor expressed in Xenopus laevis oocytes assessed as potentiation of of GABA EC5-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50240512(osthole | 7-Methoxy-8-(3-methyl-but-2-enyl)-chrome...)
Affinity DataEC50:  1.40E+4nMAssay Description:Positive allosteric modulation of human GABA-A alpha1beta2gamma2S receptor expressed in Xenopus laevis oocytes assessed as increase in GABA-induced c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50361376(OXYPEUCEDANIN)
Affinity DataEC50:  2.50E+4nMAssay Description:Positive allosteric modulation of human GABA-A alpha1beta2gamma2S receptor expressed in Xenopus laevis oocytes assessed as increase in GABA-induced c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50512168(CHEMBL4464551)
Affinity DataEC50:  9.30E+3nMAssay Description:Positive allosteric modulation of human recombinant GABA-A alpha1beta2gamma2L receptor expressed in Xenopus laevis oocytes by two-electrode voltage c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50129952(cid_5281600 | CHEMBL63354 | 8-[5-(5,7-Dihydroxy-4-...)
Affinity DataEC50:  3.60E+3nMAssay Description:Effective concentration against human recombinant GABA-A receptor alpha-1-beta-2-gamma-2 subunits expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50243877((1R,2S)-2-(aminomethyl)cyclopropanecarboxylic acid...)
Affinity DataEC50:  4.00E+4nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087271(4-Amino-but-2-enoic acid | (E)-4-Amino-but-2-enoic...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM23183(CHEMBL273481 | Muscimol | 5-(aminomethyl)-1,2-oxaz...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50243927((1S,2S)-2-(aminomethyl)cyclopropanecarboxylic acid...)
Affinity DataEC50:  5.90E+4nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50243926((1R,2R)-2-(aminomethyl)cyclopropanecarboxylic acid...)
Affinity DataEC50:  9.00E+3nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | cid_119 | Gamma-A...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGamma-aminobutyric acid type B receptor subunit 1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | cid_119 | Gamma-A...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GABAb 1A/2 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGamma-aminobutyric acid type B receptor subunit 1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50243874((+)-(S)-4-Amino-1-cyclopent-1-enyl(methyl)phosphin...)
Affinity DataEC50:  5.22E+4nMAssay Description:Agonist activity at human GABAb 1A/2 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50243873((-)-(R)-4-Amino-1-cyclopent-1-enyl(methyl)phosphin...)
Affinity DataEC50:  7.19E+4nMAssay Description:Agonist activity at human GABAb 1A/2 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50243872((+/-)-4-Amino-1-cyclopent-1-enyl(methyl)phosphinic...)
Affinity DataEC50:  5.10E+4nMAssay Description:Agonist activity at human GABAb 1A/2 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50211642(methyl(1,2,3,6-tetrahydropyridin-4-yl)phosphinic a...)
Affinity DataEC50:  5.00E+5nMAssay Description:Agonist activity at human GABAb 1A/2 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087277(4-aminobut-2-enoic acid | (Z)-4-aminobut-2-enoic a...)
Affinity DataEC50:  7.40E+4nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087269((trans)-2-Aminomethyl-cyclopropanecarboxylic acid ...)
Affinity DataEC50:  1.75E+4nMAssay Description:Partial agonist activity with low efficacy against rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087271(4-Amino-but-2-enoic acid | (E)-4-Amino-but-2-enoic...)
Affinity DataEC50:  440nMAssay Description:Partial agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087269((trans)-2-Aminomethyl-cyclopropanecarboxylic acid ...)
Affinity DataEC50:  6.80E+4nMAssay Description:Full agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM23183(CHEMBL273481 | Muscimol | 5-(aminomethyl)-1,2-oxaz...)
Affinity DataKd:  2.30E+3nMAssay Description:Partial agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087271(4-Amino-but-2-enoic acid | (E)-4-Amino-but-2-enoic...)
Affinity DataEC50:  600nMAssay Description:Partial agonist activity against homomeric rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087269((trans)-2-Aminomethyl-cyclopropanecarboxylic acid ...)
Affinity DataEC50:  2.00E+4nMAssay Description:Full agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087273(4-Amino-2-fluoro-but-2-enoic acid (2-FTACA) | CHEM...)
Affinity DataEC50:  2.43E+3nMAssay Description:Partial agonist activity against rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087269((trans)-2-Aminomethyl-cyclopropanecarboxylic acid ...)
Affinity DataEC50:  3.45E+4nMAssay Description:Full agonist activity against human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087274(4-amino-2-methylbut-2-enoic acid | 4-Amino-2-methy...)
Affinity DataEC50:  1.01E+5nMAssay Description:Activation of human rho2 GABA-C receptor at 34% of maximal GABA-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM85712(1H-imidazol-4-ylacetic acid | NSC_96215 | CAS_645-...)
Affinity DataEC50:  1.60E+4nMAssay Description:Partial agonist activity against rho-1 subunit GABA-C receptor expressed in Xenopus oocytes, low intrinsic activity (Im 3%)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087276(3-Amino-propane-1-sulfinic acid (Homohypotaurine) ...)
Affinity DataEC50:  4.60E+3nMAssay Description:Partial agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM23183(CHEMBL273481 | Muscimol | 5-(aminomethyl)-1,2-oxaz...)
Affinity DataKd:  1.40E+3nMAssay Description:Partial agonist activity against human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087277(4-aminobut-2-enoic acid | (Z)-4-aminobut-2-enoic a...)
Affinity DataEC50:  7.00E+4nMAssay Description:Partial agonist activity against human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087271(4-Amino-but-2-enoic acid | (E)-4-Amino-but-2-enoic...)
Affinity DataEC50:  400nMAssay Description:Partial agonist activity against homomeric rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50087277(4-aminobut-2-enoic acid | (Z)-4-aminobut-2-enoic a...)
Affinity DataEC50:  7.40E+4nMAssay Description:Partial agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM85712(1H-imidazol-4-ylacetic acid | NSC_96215 | CAS_645-...)
Affinity DataEC50:  3.00E+3nMAssay Description:Partial agonist activity against human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50374647(CHEMBL256608)
Affinity DataEC50:  6.50E+4nMAssay Description:Agonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50021187(R(-)-4-amino-3-hydroxybutanoic acid | CHEMBL290216...)
Affinity DataEC50:  1.91E+4nMAssay Description:Agonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | cid_119 | Gamma-A...)
Affinity DataEC50:  1.19E+3nMAssay Description:Agonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50021186(CHEMBL296263 | S(+)-4-amino-3-hydroxybutanoic acid...)
Affinity DataEC50:  4.48E+4nMAssay Description:Agonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50374648(CHEMBL403157)
Affinity DataEC50:  4.00E+4nMAssay Description:Agonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50300802(CHEMBL1084615 | CHEMBL565540 | 5-Morpholin-4-ylpen...)
Affinity DataEC50:  1.65E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50300802(CHEMBL1084615 | CHEMBL565540 | 5-Morpholin-4-ylpen...)
Affinity DataEC50:  9.50E+3nMAssay Description:Partial agonist activity at wild type rat recombinant alpha7 nAChR expressed in Xenopus oocyte by voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50300811(N-{4-[4-(2,4-dimethoxyphenyl)-piperazin-1-yl]butyl...)
Affinity DataEC50:  2.84E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in HEK292 cells after 4 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM23183(CHEMBL273481 | Muscimol | 5-(aminomethyl)-1,2-oxaz...)
Affinity DataEC50:  2.30E+3nMAssay Description:Partial agonist activity at GABAC rho1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50218536(4(5)-(carboxymethyl)-5(4)-methylimidazole | CHEMBL...)
Affinity DataEC50:  2.20E+4nMAssay Description:Agonist activity at GABAC rho1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50241194((1S,2R)-2-aminomethyl-cyclopropanecarboxylic acid ...)
Affinity DataEC50:  3.97E+4nMAssay Description:Agonist activity at GABAC rho1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | cid_119 | Gamma-A...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at GABAC rho1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587468(CHEMBL2296158)
Affinity DataIC50: 90nMAssay Description:Inhibition of human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587468(CHEMBL2296158)
Affinity DataIC50: 90nMAssay Description:Inhibition of human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
Displayed 1 to 50 (of 159 total ) | Next | Last >>
Jump to: