Compile Data Set for Download or QSAR
Found 1176 with Last Name = 'chung' and Initial = 's'
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50366620(RESINIFERATOXIN)
Affinity DataKi:  0.0426nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247744(CHEMBL504725 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  0.0730nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Jilin University

Curated by ChEMBL
LigandPNGBDBM50483252(CHEMBL1643369)
Affinity DataKi:  0.200nMAssay Description:Inhibition of Escherichia coli LpxCMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Jilin University

Curated by ChEMBL
LigandPNGBDBM50483252(CHEMBL1643369)
Affinity DataKi:  0.200nMAssay Description:Inhibition of Escherichia coli LpxCMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247741(CHEMBL503101 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  0.228nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247749(CHEMBL510583 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Jilin University

Curated by ChEMBL
LigandPNGBDBM92267(CS257)
Affinity DataKi:  0.550nMAssay Description:Inhibition of Escherichia coli LpxCMore data for this Ligand-Target Pair
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Escherichia coli)
Jilin University

Curated by ChEMBL
LigandPNGBDBM92267(CS257)
Affinity DataKi:  0.550nMAssay Description:Inhibition of Escherichia coli LpxCMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247742(CHEMBL509154 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247748(CHEMBL510228 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247751(CHEMBL449201 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  0.980nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284388(2-{[Acetyl-(1-hexadecylcarbamoyloxymethyl-cyclopen...)
Affinity DataKi:  1.20nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247745(CHEMBL455555 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247750(CHEMBL455155 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  2.69nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247746(CHEMBL502769 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247747(CHEMBL509331 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  3.53nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284401(2-{[Acetyl-(1-octadecylcarbamoyloxymethyl-cyclopen...)
Affinity DataKi:  4.20nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284416(2-{[Acetyl-(3-octadecylcarbamoyloxymethyl-cyclobut...)
Affinity DataKi:  4.30nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284419(2-{[Acetyl-((2R,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataKi:  4.30nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284417(2-{[Acetyl-((2R,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataKi:  5.70nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284395(2-{[Acetyl-(1-octadecylcarbamoyloxymethyl-cyclobut...)
Affinity DataKi:  6.60nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247743(CHEMBL504206 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  6.81nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataKi:  7.20nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataKi:  7.20nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50247752(CHEMBL462654 | [(1R,2R,6R,10S,11R,15S,17R)-13-benz...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]RTX form rat TRPV1 receptor expressed in CHO/VR1 cell systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284414(2-{[Acetyl-((2S,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataKi:  9.20nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284399(1-[4-(1-Octadecylcarbamoyloxymethyl-cyclopentylmet...)
Affinity DataKi:  9.40nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284412(2-{[Acetyl-((2S,4S)-4-hexadecylcarbamoyloxymethyl-...)
Affinity DataKi:  9.80nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284420(2-{[Acetyl-((2S,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataKi:  9.80nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284409(2-{[Acetyl-(2,2-dimethyl-3-octadecylcarbamoyloxy-p...)
Affinity DataKi:  13nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284414(2-{[Acetyl-((2S,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataKi:  15nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284422(2-{[Acetyl-((2S,4S)-4-hexadecyloxymethyl-oxetan-2-...)
Affinity DataKi:  15nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284400(2-{[Acetyl-(3-octadecylcarbamoyloxymethyl-oxetan-3...)
Affinity DataKi:  20nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284423(2-{[Acetyl-((2R,4R)-4-hexadecyloxymethyl-thietan-2...)
Affinity DataKi:  20nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284386(1-[5-(3-Octadecylcarbamoyloxymethyl-thietan-3-ylme...)
Affinity DataKi:  20nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetFatty acid-binding protein, liver(Mus musculus (Mouse))
Avanti Polar Lipids

LigandPNGBDBM50212873(((2'-(5-ETHYL-3,4-DIPHENYL-1H-PYRAZOL-1-YL)-3-BIPH...)
Affinity DataKi:  21nMAssay Description:The following fluorescent ligand displacement assays at 24 °C were used to further confirm and/or determine if the cytosolic lipidic ligand "chaperon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284413(2-{[Acetyl-((2S,4R)-4-hexadecyloxymethyl-oxetan-2-...)
Affinity DataKi:  21nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284400(2-{[Acetyl-(3-octadecylcarbamoyloxymethyl-oxetan-3...)
Affinity DataKi:  23nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20287(2-[(4-tert-butylphenyl)methyl]-3-({[(3-fluoro-4-me...)
Affinity DataKi:  23nMAssay Description:Binding affinity towards rat vanilloid receptor subtype 1 expressed in CHO cells by [3H]-RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytidine deaminase(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50367034(CHEMBL610997)
Affinity DataKi:  25nMAssay Description:Binding affinity for human cytidine deaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284415(1-Ethyl-2-{[((2R,4R)-4-hexadecylcarbamoyloxymethyl...)
Affinity DataKi:  26nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284398(3-[5-(3-Octadecylcarbamoyloxymethyl-thietan-3-ylme...)
Affinity DataKi:  28nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50130542(2,2-Dimethyl-propionic acid 2-(3,4-dimethyl-benzyl...)
Affinity DataKi:  29nMAssay Description:Agonist effect on 45 [Ca2+] influx in vanilloid receptor expressing CHO cells relative to maximal capsaicin (300 nM) response, weak effect at 30 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty acid-binding protein, liver(Mus musculus (Mouse))
Avanti Polar Lipids

LigandPNGBDBM50054471((5Z,8Z)-Icosa-5,8,11,14-tetraenoic acid (4-hydroxy...)
Affinity DataKi:  29nMAssay Description:The following fluorescent ligand displacement assays at 24 °C were used to further confirm and/or determine if the cytosolic lipidic ligand "chaperon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284392(1-[5-(3-Octadecylcarbamoyloxymethyl-thietan-3-ylme...)
Affinity DataKi:  30nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284396(3-[5-(3-Octadecylcarbamoyloxymethyl-oxetan-3-ylmet...)
Affinity DataKi:  31nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetFatty acid-binding protein, liver(Mus musculus (Mouse))
Avanti Polar Lipids

LigandPNGBDBM197171(4,4,8-trimethyl-5-(3-methylbutanoyl)-4,5-dihydro-1...)
Affinity DataKi:  33nMAssay Description:The following fluorescent ligand displacement assays at 24 °C were used to further confirm and/or determine if the cytosolic lipidic ligand "chaperon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284410(1-Ethyl-2-{[(4-methoxy-benzoyl)-(4-octadecylcarbam...)
Affinity DataKi:  34nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284411(2-{[Acetyl-((2R,4R)-1-acetyl-4-octadecylcarbamoylo...)
Affinity DataKi:  35nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetFatty acid-binding protein, liver(Mus musculus (Mouse))
Avanti Polar Lipids

LigandPNGBDBM197167(N-(4-hydroxy-2-methylphenyl)icosa-5,8,11,14-tetrae...)
Affinity DataKi:  37nMAssay Description:The following fluorescent ligand displacement assays at 24 °C were used to further confirm and/or determine if the cytosolic lipidic ligand "chaperon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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