Compile Data Set for Download or QSAR
Report error Found 290 with Last Name = 'clerin' and Initial = 'v'
TargetAtypical chemokine receptor 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50264279(CHEMBL4072602)
Affinity DataEC50:  7nMAssay Description:Modulation of prolink-tagged human CXCR7 expressed in CHO-K1 cells assessed as induction of beta-arrestin recruitment after 30 mins by beta-galactosi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50264280(CHEMBL4084050)
Affinity DataEC50:  11nMAssay Description:Modulation of prolink-tagged human CXCR7 expressed in CHO-K1 cells assessed as induction of beta-arrestin recruitment after 30 mins by beta-galactosi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20015(2-[4-({[3-(3-benzyl-8-chloroquinolin-4-yl)phenyl]a...)
Affinity DataIC50: 1.40nM EC50:  23nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20024(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 1.40nM EC50:  316nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20001(2-{4-[({3-[3-benzyl-8-(trifluoromethyl)quinolin-4-...)
Affinity DataIC50: 1.90nM EC50:  33nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20001(2-{4-[({3-[3-benzyl-8-(trifluoromethyl)quinolin-4-...)
Affinity DataIC50: 1.90nM EC50:  33nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20000(CHEMBL214719 | 2-(4-{3-[3-benzyl-8-(trifluoromethy...)
Affinity DataIC50: 2nM EC50:  90nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20001(2-{4-[({3-[3-benzyl-8-(trifluoromethyl)quinolin-4-...)
Affinity DataIC50: 2nM EC50:  90nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20000(CHEMBL214719 | 2-(4-{3-[3-benzyl-8-(trifluoromethy...)
Affinity DataIC50: 2.10nM EC50:  71nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20004(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 2.40nM EC50:  29nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20020(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 2.60nM EC50:  58nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20014(2-[4-({[3-(3-benzoyl-8-chloroquinolin-4-yl)phenyl]...)
Affinity DataIC50: 2.70nM EC50:  39nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20006(2-{4-[({3-[3-phenyl-8-(trifluoromethyl)quinolin-4-...)
Affinity DataIC50: 3.70nM EC50:  44nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20021(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 3.80nM EC50:  78nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20005(2-{4-[({3-[3-methyl-8-(trifluoromethyl)quinolin-4-...)
Affinity DataIC50: 4.30nM EC50:  100nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM19999(2-(4-{3-[3-benzoyl-8-(trifluoromethyl)quinolin-4-y...)
Affinity DataIC50: 5nM EC50:  143nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20015(2-[4-({[3-(3-benzyl-8-chloroquinolin-4-yl)phenyl]a...)
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20011(2-[4-({[3-(3-benzyl-8-methylquinolin-4-yl)phenyl]a...)
Affinity DataIC50: 5nM EC50:  90nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20025(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 5.40nM EC50:  795nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20010(2-[4-({[3-(3-benzoyl-8-methylquinolin-4-yl)phenyl]...)
Affinity DataIC50: 5.5nM EC50:  61nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20016(2-{3-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 6nM EC50:  141nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20002(CHEMBL216645 | 2-{4-[({3-[3-benzyl-8-(trifluoromet...)
Affinity DataIC50: 7nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20004(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 7nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20001(2-{4-[({3-[3-benzyl-8-(trifluoromethyl)quinolin-4-...)
Affinity DataIC50: 7.60nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20001(2-{4-[({3-[3-benzyl-8-(trifluoromethyl)quinolin-4-...)
Affinity DataIC50: 7.60nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20023(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 7.80nM EC50:  2.40E+3nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20006(2-{4-[({3-[3-phenyl-8-(trifluoromethyl)quinolin-4-...)
Affinity DataIC50: 8nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20001(2-{4-[({3-[3-benzyl-8-(trifluoromethyl)quinolin-4-...)
Affinity DataIC50: 8nM EC50:  160nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20022(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 8.5nM EC50:  4.00E+3nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20014(2-[4-({[3-(3-benzoyl-8-chloroquinolin-4-yl)phenyl]...)
Affinity DataIC50: 9nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataIC50: 9nM EC50:  170nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20000(CHEMBL214719 | 2-(4-{3-[3-benzyl-8-(trifluoromethy...)
Affinity DataIC50: 9.5nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataIC50: 10nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataIC50: 10nM EC50:  16nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM26065(2-[(2,4-dimethylphenyl)methyl]-3-(4-fluorophenyl)-...)
Affinity DataIC50: 10nM EC50:  990nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20000(CHEMBL214719 | 2-(4-{3-[3-benzyl-8-(trifluoromethy...)
Affinity DataIC50: 10nM EC50:  240nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20024(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 11nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM19992(2-{3-[3-({[2-chloro-3-(trifluoromethyl)phenyl]meth...)
Affinity DataIC50: 12nM EC50:  410nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20017(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 12nM EC50:  1.27E+3nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM19992(2-{3-[3-({[2-chloro-3-(trifluoromethyl)phenyl]meth...)
Affinity DataIC50: 12nM EC50:  310nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20027({4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4-y...)
Affinity DataIC50: 12.8nM EC50:  2.30E+3nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataIC50: 13nM EC50:  140nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20020(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 15.2nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20005(2-{4-[({3-[3-methyl-8-(trifluoromethyl)quinolin-4-...)
Affinity DataIC50: 16nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM19999(2-(4-{3-[3-benzoyl-8-(trifluoromethyl)quinolin-4-y...)
Affinity DataIC50: 16.5nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM20012(2-[4-({[3-(3-benzoyl-8-fluoroquinolin-4-yl)phenyl]...)
Affinity DataIC50: 17nM EC50:  700nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20021(2-{4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4...)
Affinity DataIC50: 17.2nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20010(2-[4-({[3-(3-benzoyl-8-methylquinolin-4-yl)phenyl]...)
Affinity DataIC50: 18nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-alpha [197-447](Human)
Wyeth Research

LigandPNGBDBM20011(2-[4-({[3-(3-benzyl-8-methylquinolin-4-yl)phenyl]a...)
Affinity DataIC50: 21nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetOxysterols receptor LXR-beta [154-461](Human)
Wyeth Research

LigandPNGBDBM26066(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
Affinity DataIC50: 24nM EC50:  3.67E+3nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 290 total ) | Next | Last >>
Jump to: