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TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataKi:  5nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataKi:  6nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataKi:  6nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121622(4-[2-(4-(4-Benzyl-piperazin-1-yl)-6-{[3-(4-chloro-...)
Affinity DataKi:  8nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121590(4-{2-[4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121626(4-(2-{4-[3-(4-Chloro-phenyl)-propylsulfanyl]-6-pip...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121602(4-[2-(4-{[3-(4-Fluoro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121589(4-(2-{4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121598(4-{2-[4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121608(4-[2-(4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143827((E)-3-[4-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,8-te...)
Affinity DataKi:  20nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143825(5-[1-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-na...)
Affinity DataKi:  20nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121584(4-[2-(4-{[3-(3,4-Difluoro-phenyl)-propyl]-methyl-a...)
Affinity DataKi:  20nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121601(4-[2-(4-{[3-(2,4-Dichloro-phenyl)-propyl]-methyl-a...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121604(4-(2-{4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121634(4-[2-(4-(4-Allyl-piperazin-1-yl)-6-{[3-(4-chloro-p...)
Affinity DataKi:  30nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121603(4-(2-{4-[(3-Benzo[1,3]dioxol-5-yl-propyl)-methyl-a...)
Affinity DataKi:  30nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121600(4-{2-[4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  35nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121636(1-(4-{4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  40nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121633(4-[2-(4-{[3-(2-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  40nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143833((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataKi:  40nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121625(4-{2-[4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  40nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121587(CHEMBL153395 | cis-4-(2-{4-[Methyl-(2-phenyl-cyclo...)
Affinity DataKi:  40nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143832((E)-3-[4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro...)
Affinity DataKi:  40nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121588(4-{2-[4-(4-Methyl-piperazin-1-yl)-6-(3-phenyl-prop...)
Affinity DataKi:  50nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121593(4-{2-[4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  50nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121596(4-(2-{4-[3-(4-Chloro-phenyl)-propylamino]-6-pipera...)
Affinity DataKi:  55nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121590(4-{2-[4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  60nMAssay Description:In vitro binding affinity towards human Estrogen receptor alpha using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50409928(CHEMBL2113737)
Affinity DataKi:  63nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121594(4-[2-(4-{Methyl-[3-(4-trifluoromethyl-phenyl)-prop...)
Affinity DataKi:  75nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50409929(CHEMBL2113736)
Affinity DataKi:  79nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataKi:  90nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121620(4-[3-({4-[2-(4-Hydroxy-phenyl)-ethylamino]-6-piper...)
Affinity DataKi:  90nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121607(4-(2-{4-[2-(4-Chloro-phenoxy)-ethylsulfanyl]-6-pip...)
Affinity DataKi:  90nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143824((E)-3-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataKi:  93nMAssay Description:Binding affinity for retinoic acid receptor alpha (RARalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121632(1-(4-{4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  100nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121613(4-(2-{4-[Methyl-(3-p-tolyl-propyl)-amino]-6-pipera...)
Affinity DataKi:  100nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143821((E)-3-[4-(5,5,8,8-Tetramethyl-3-propoxy-5,6,7,8-te...)
Affinity DataKi:  100nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121624(4-[2-(4-{[3-(4-Chloro-phenyl)-propyl]-ethyl-amino}...)
Affinity DataKi:  100nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121609((4-{4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino}-...)
Affinity DataKi:  110nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121614(1-(4-{4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  110nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121621(4-{2-[4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  115nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121622(4-[2-(4-(4-Benzyl-piperazin-1-yl)-6-{[3-(4-chloro-...)
Affinity DataKi:  120nMAssay Description:In vitro binding affinity towards human Estrogen receptor alpha using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121601(4-[2-(4-{[3-(2,4-Dichloro-phenyl)-propyl]-methyl-a...)
Affinity DataKi:  125nMAssay Description:In vitro binding affinity towards human Estrogen receptor alpha using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143835((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataKi:  138nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121598(4-{2-[4-{[3-(4-Chloro-phenyl)-propyl]-methyl-amino...)
Affinity DataKi:  145nMAssay Description:In vitro binding affinity towards human Estrogen receptor alpha using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143823((E)-3-[5-Methyl-4-(5,5,8,8-tetramethyl-5,6,7,8-tet...)
Affinity DataKi:  158nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143831((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataKi:  158nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121626(4-(2-{4-[3-(4-Chloro-phenyl)-propylsulfanyl]-6-pip...)
Affinity DataKi:  160nMAssay Description:In vitro binding affinity towards human Estrogen receptor alpha using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50121610(4-[2-(4-{[2-(4-Chloro-phenoxy)-ethyl]-methyl-amino...)
Affinity DataKi:  170nMAssay Description:In vitro binding affinity towards human Estrogen receptor 2 using [3H]-17-beta-estradiol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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