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TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023394((4-{1-[2-(4-Azido-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  2.86E+3nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of [125-I]-labeled aminobenzyl adenosine binding to bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023391({4-[1-(4-Amino-3-iodo-benzyl)-2,6-dioxo-3-propyl-2...)
Affinity DataKd:  160nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50008405(CHEMBL27041 | 2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7...)
Affinity DataKd:  17nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of [125-I]-labeled aminobenzyl adenosine binding to bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023392({4-[3-(4-Amino-benzyl)-2,6-dioxo-1-propyl-2,3,6,9-...)
Affinity DataKd:  32nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023396((4-{3-[2-(4-Amino-phenyl)-ethyl]-2,6-dioxo-1-propy...)
Affinity DataKd:  60nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82558(NSC_163889 | CAS_163889 | CHEMBL355370 | I-ABOPX)
Affinity DataKd:  37nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023400((4-{1,3-Bis-[2-(4-amino-phenyl)-ethyl]-2,6-dioxo-2...)
Affinity DataKd:  3.59E+3nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023401((4-{1-[2-(4-Amino-phenyl)-ethyl]-2,6-dioxo-3-propy...)
Affinity DataKd:  2.30E+3nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023395((4-{3-[2-(4-Azido-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  24nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023398((4-{3-[2-(4-Amino-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  29nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023390({4-[1-(4-Amino-benzyl)-2,6-dioxo-3-propyl-2,3,6,9-...)
Affinity DataKd:  44nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023397({4-[1-(4-Azido-3-iodo-benzyl)-2,6-dioxo-3-propyl-2...)
Affinity DataKd:  960nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of [125-I]-labeled aminobenzyl adenosine binding to bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023399({4-[3-(4-Azido-3-iodo-benzyl)-2,6-dioxo-1-propyl-2...)
Affinity DataKd:  55nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of [125-I]-labeled aminobenzyl adenosine binding to bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023395((4-{3-[2-(4-Azido-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  1.20nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain membrane(KD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023398((4-{3-[2-(4-Amino-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  0.800nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain membrane(KD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82558(NSC_163889 | CAS_163889 | CHEMBL355370 | I-ABOPX)
Affinity DataKd:  0.800nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain membrane(KD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023402((4-{1-[2-(4-Amino-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  3.10E+3nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataIC50: 0.350nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50367678(CHEMBL605469)
Affinity DataIC50: 0.900nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 2.40nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82558(NSC_163889 | CAS_163889 | CHEMBL355370 | I-ABOPX)
Affinity DataIC50: 3nMAssay Description:Binding affinity towards adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82558(NSC_163889 | CAS_163889 | CHEMBL355370 | I-ABOPX)
Affinity DataIC50: 3nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023392({4-[3-(4-Amino-benzyl)-2,6-dioxo-1-propyl-2,3,6,9-...)
Affinity DataIC50: 3.40nMAssay Description:Binding affinity towards adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023390({4-[1-(4-Amino-benzyl)-2,6-dioxo-3-propyl-2,3,6,9-...)
Affinity DataIC50: 5.20nMAssay Description:Binding affinity towards adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82015(1,3-Dimethyl-8-phenyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataIC50: 8.80nMAssay Description:Binding affinity towards adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023396((4-{3-[2-(4-Amino-phenyl)-ethyl]-2,6-dioxo-1-propy...)
Affinity DataIC50: 16nMAssay Description:Inhibition of photolabeling of 34 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82015(1,3-Dimethyl-8-phenyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataIC50: 18nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM81971(1,3-Diethyl-8-phenyl-3,7-dihydro-purine-2,6-dione ...)
Affinity DataIC50: 32nMAssay Description:Binding affinity towards adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023396((4-{3-[2-(4-Amino-phenyl)-ethyl]-2,6-dioxo-1-propy...)
Affinity DataIC50: 37nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023396((4-{3-[2-(4-Amino-phenyl)-ethyl]-2,6-dioxo-1-propy...)
Affinity DataIC50: 37nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023390({4-[1-(4-Amino-benzyl)-2,6-dioxo-3-propyl-2,3,6,9-...)
Affinity DataIC50: 44nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM81971(1,3-Diethyl-8-phenyl-3,7-dihydro-purine-2,6-dione ...)
Affinity DataIC50: 48nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023392({4-[3-(4-Amino-benzyl)-2,6-dioxo-1-propyl-2,3,6,9-...)
Affinity DataIC50: 64nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50367678(CHEMBL605469)
Affinity DataIC50: 430nMAssay Description:Inhibition of photolabeling of 34 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataIC50: 720nMAssay Description:Binding affinity towards adenosine A1 receptor rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50367678(CHEMBL605469)
Affinity DataIC50: 1.15E+3nMAssay Description:Binding affinity towards adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 2.46E+3nMAssay Description:Binding affinity towards adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of photolabeling of 34 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of photolabeling of 24 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of photolabeling of 34 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of photolabeling of 24 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82558(NSC_163889 | CAS_163889 | CHEMBL355370 | I-ABOPX)
Affinity DataKi:  700nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50008405(CHEMBL27041 | 2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7...)
Affinity DataKi:  800nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023392({4-[3-(4-Amino-benzyl)-2,6-dioxo-1-propyl-2,3,6,9-...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023391({4-[1-(4-Amino-3-iodo-benzyl)-2,6-dioxo-3-propyl-2...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023399({4-[3-(4-Azido-3-iodo-benzyl)-2,6-dioxo-1-propyl-2...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023398((4-{3-[2-(4-Amino-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023397({4-[1-(4-Azido-3-iodo-benzyl)-2,6-dioxo-3-propyl-2...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023395((4-{3-[2-(4-Azido-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKi:  5.40E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023396((4-{3-[2-(4-Amino-phenyl)-ethyl]-2,6-dioxo-1-propy...)
Affinity DataKi:  1.15E+4nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
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