Report error Found 1669 with Last Name = 'dai' and Initial = 'j'
Affinity DataKi: 1.20nMAssay Description:Displacement of [125I-HEAT from human alpha1D-adrenoreceptor expressed in CHOK1 cell membranes incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Competitive inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using ATP as subst...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [125I-HEAT from human alpha1A-adrenoreceptor expressed in CHOK1 cell membranes incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Competitive inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using ATP as subst...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataKi: 7.60nMAssay Description:Competitive inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using ATP as subst...More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Competitive inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using ATP as subst...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [125I]BOB-4 from Amyloid beta (1 to 42) (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Competitive inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using ATP as subst...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of LSD1 (unknown origin) assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Mean functional activity against human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [125I-HEAT from human alpha1B-adrenoreceptor expressed in CHOK1 cell membranes incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [125I]BOB-4 from Amyloid beta (1 to 42) (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [125I]BOB-4 from Amyloid beta (1 to 42) (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [125I]BOB-4 from Amyloid beta (1 to 42) (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [125I]BOB-4 from Amyloid beta (1 to 42) (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Blocking activity was assessed by antagonism of (-)-noradrenaline induced contraction of rat prostatic vas deferens (alpha1A adrenoceptor)More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Mean functional activity against human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [125I]1-Iodo-4-((4-methoxyphenoxy)methyl)benzene from amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
