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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataEC50:  200nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29078(cyclopropanolamide, 13a | racemic | cyclopropanola...)
Affinity DataEC50:  1.90E+3nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29079(cyclopropanolamide, 12a | racemic | cyclopropanola...)
Affinity DataEC50:  50nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29080(Oleamide MEA | Oleoyl monoethanolamide | CHEMBL280...)
Affinity DataEC50:  3.65E+3nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29081(cyclopropanolamide, 13b | racemic | cyclopropanola...)
Affinity DataEC50:  3.70E+3nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29082(cyclopropanolamide, 12b | racemic | cyclopropanola...)
Affinity DataEC50:  60nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29083(Palmidrol | Impulsin | MimyX | Palmityoletanolamid...)
Affinity DataEC50: >1.00E+4nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29084(racemic | cyclopropanolamide, rac-10c)
Affinity DataEC50:  2.64E+4nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29085(cyclopropanolamide, rac-9c)
Affinity DataEC50:  40nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataEC50:  20nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29078(cyclopropanolamide, 13a | racemic | cyclopropanola...)
Affinity DataEC50:  610nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29087(cyclopropanolamide, 14a)
Affinity DataEC50:  2.40E+3nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29088(cyclopropanolamide, 11a)
Affinity DataEC50:  47nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29079(cyclopropanolamide, 12a | racemic | cyclopropanola...)
Affinity DataEC50:  23nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29081(cyclopropanolamide, 13b | racemic | cyclopropanola...)
Affinity DataEC50:  150nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29091(cyclopropanolamide, 14b)
Affinity DataEC50:  180nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29082(cyclopropanolamide, 12b | racemic | cyclopropanola...)
Affinity DataEC50:  13nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29093(cyclopropanolamide, 11b)
Affinity DataEC50:  19nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  565nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB1 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluorescence as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  73nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB2 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  1.61E+4nMAssay Description:Agonist activity at recombinant rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  7.30E+3nMAssay Description:Agonist activity at recombinant rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at recombinant rat TRPV3 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  75nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB1 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  4.78E+3nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB2 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  200nMAssay Description:Agonist activity at recombinant rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  6.20E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluorescence as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  180nMAssay Description:Agonist activity at recombinant rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  5.30E+3nMAssay Description:Agonist activity at recombinant rat TRPV3 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463445(CHEMBL4238545)
Affinity DataEC50:  490nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM50463442(CHEMBL4242719)
Affinity DataEC50:  4.90E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463442(CHEMBL4242719)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463443(CHEMBL4241477)
Affinity DataEC50:  350nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463447(CHEMBL4249046)
Affinity DataEC50:  6.70E+3nMAssay Description:Agonist activity at rat TRPV3 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463442(CHEMBL4242719)
Affinity DataEC50:  6.40E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463447(CHEMBL4249046)
Affinity DataEC50:  5.80E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463446(CHEMBL4244422)
Affinity DataEC50:  8.40E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM50463445(CHEMBL4238545)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM50463447(CHEMBL4249046)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463446(CHEMBL4244422)
Affinity DataEC50:  230nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463447(CHEMBL4249046)
Affinity DataEC50:  290nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463444(CHEMBL4238978)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463445(CHEMBL4238545)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463443(CHEMBL4241477)
Affinity DataEC50:  1.80E+4nMAssay Description:Agonist activity at rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463445(CHEMBL4238545)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM50278349(2-(Diphenylboryloxy)Ethanamine | 2-Aminoethoxydiph...)
Affinity DataEC50:  1.29E+5nMAssay Description:Agonist activity at recombinant human TRPV1 expressed in HEK293 cells assessed as induction of Ca2+ levels by Fuo-4-AM based spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM50473840(CHEMBL122039)
Affinity DataEC50:  79nMAssay Description:Concentration necessary to induce a relative half-maximal response measured by the entry of [Ca2+] into human embryonic kidney HEK293 cells overexpre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
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