Compile Data Set for Download or QSAR
Report error Found 49 with Last Name = 'diel' and Initial = 'pj'
LigandPNGBDBM24184((3-aminopropyl)phosphinic acid | CHEMBL112203 | CG...)
Affinity DataIC50: 5nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM24185(CGP35024 | 3-Apmpa | CHEMBL112710 | (3-aminopropyl...)
Affinity DataIC50: 16nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50033007((3-Amino-propyl)-(3-oxo-butyl)-phosphinic acid | C...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032996((3-Amino-propyl)-[2-(tetrahydro-pyran-2-yl)-ethyl]...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033008((3-Amino-propyl)-[3-(2-carbamoyl-benzoylamino)-2-h...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032972(CGP-36216 | (3-Amino-propyl)-ethyl-phosphinic acid...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033024((3-Amino-propyl)-(2-cyclohexyl-ethyl)-phosphinic a...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033017((3-Amino-propyl)-cyclohexylmethyl-phosphinic acid ...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032989(CHEMBL113308 | CHEMBL112019 | ((S)-3-Amino-2-hydro...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032989(CHEMBL113308 | CHEMBL112019 | ((S)-3-Amino-2-hydro...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033014(((R)-3-Amino-2-hydroxy-propyl)-benzyl-phosphinic a...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032987((3-Amino-propyl)-pyridin-2-ylmethyl-phosphinic aci...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032984([3-Amino-2-(4-chloro-phenyl)-2-hydroxy-propyl]-met...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032989(CHEMBL113308 | CHEMBL112019 | ((S)-3-Amino-2-hydro...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033004([3-Amino-2-(4-chloro-phenyl)-2-hydroxy-propyl]-but...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033014(((R)-3-Amino-2-hydroxy-propyl)-benzyl-phosphinic a...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033016((3-Amino-propyl)-(hydroxy-phenyl-methyl)-phosphini...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033011([3-Amino-2-(4-chloro-phenyl)-propyl]-methyl-phosph...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033029((3-Amino-propyl)-phenethyl-phosphinic acid | CHEMB...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033018((3-Amino-propyl)-benzyl-phosphinic acid | CHEMBL11...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032997(CHEMBL324244 | ((S)-3-Amino-2-hydroxy-propyl)-diet...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032995((3-Amino-2-oxo-propyl)-cyclopropylmethyl-phosphini...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032990((3-Amino-propyl)-isobutyl-phosphinic acid | CHEMBL...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033013((3-Amino-propyl)-propyl-phosphinic acid | CHEMBL11...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032997(CHEMBL324244 | ((S)-3-Amino-2-hydroxy-propyl)-diet...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032994((3-Amino-propyl)-(1-hydroxy-butyl)-phosphinic acid...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033019((3-Amino-propyl)-diisopropoxymethyl-phosphinic aci...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033027((3-Amino-propyl)-hexyl-phosphinic acid | CHEMBL113...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033021((3-Amino-propyl)-dibutoxymethyl-phosphinic acid | ...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033009([3-Amino-2-(4-chloro-phenyl)-propyl]-diethoxymethy...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033012((3-Amino-propyl)-(1,1-difluoro-butyl)-phosphinic a...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033003(CGP-35348 | (3-Amino-propyl)-diethoxymethyl-phosph...)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50032986((3-Amino-propyl)-dipropoxymethyl-phosphinic acid |...)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032998((3-Amino-2-hydroxy-propyl)-butyl-phosphinic acid |...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032985(Bis-(3-amino-propyl)-phosphinic acid | CHEMBL11229...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033014(((R)-3-Amino-2-hydroxy-propyl)-benzyl-phosphinic a...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033000((3-Amino-propyl)-(tetrahydro-pyran-2-ylmethyl)-pho...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032992((3-Amino-propyl)-(tetrahydro-furan-2-yl)-phosphini...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033001((3-Amino-propyl)-cyclopropylmethyl-phosphinic acid...)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033028((3-Amino-1-hydroxy-propyl)-butyl-phosphinic acid |...)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032982(CGP36742 | 3-aminopropyl(butyl)phosphinic acid | C...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033026((3-Amino-propyl)-(tetrahydro-pyran-2-yl)-phosphini...)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032983((3-Amino-2-hydroxy-2-methyl-propyl)-butyl-phosphin...)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033023(Aminomethyl-(3-amino-propyl)-phosphinic acid | CHE...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033025((3-Amino-2-oxo-propyl)-cyclohexylmethyl-phosphinic...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033002((3-Amino-propyl)-(4-fluoro-benzyl)-phosphinic acid...)
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50033010((3-Amino-propyl)-tert-butyl-phosphinic acid | CHEM...)
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032993((3-Amino-propyl)-phenyl-phosphinic acid | CHEMBL11...)
Affinity DataIC50: 1.26E+5nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032988((3-Amino-1-methyl-propyl)-butyl-phosphinic acid | ...)
Affinity DataIC50: 3.41E+5nMAssay Description:Inhibition of binding of [3H]CGP-27492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed