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TargetProstaglandin E synthase(Human)
Bhupat and Jyoti Mehta School of Biosciences

Curated by ChEMBL
LigandPNGBDBM50038649(ML-3000 | [2-(4-Chloro-phenyl)-6,6-dimethyl-1-phen...)
Affinity DataEC50:  100nMAssay Description:Inhibition of mPGES1 in human A549 cells assessed as reduction in PGE2 productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324297(4-(1-Piperazin-1-yl[2,6]naphthyridin-3-yl)pyridin-...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324315(N-cyclohexyl-4-(1-(piperazin-1-yl)-2,6-naphthyridi...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094166(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataIC50: 0.75nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094131(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2-bromo-phenyl)-...)
Affinity DataIC50: 0.880nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469565(CHEMBL4082918)
Affinity DataIC50: 1nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC using UDP-3-O-(R-hydroxydecanoyl)-N-acetylglucosamine as substrate preincubated for 30 mins followed by sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324306(1-[3-(2-Cyclohexylaminopyridin-4-yl)[2,6]naphthyri...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324305(N-(2-(pyrrolidin-1-yl)ethyl)-1-(3-(2-(tetrahydro-2...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324296(1-[3-(2-Cyclohexylaminopyridin-4-yl)[2,6]naphthyri...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324298({4-[1-(4-Isobutylpiperazin-1-yl)[2,6]naphthyridin-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324314(1-{3-[2-(Tetrahydropyran-4-ylamino)pyridin-4-yl][2...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094178(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2-bromo-phenyl)-...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094137(N-[2-Benzo[1,3]dioxol-4-yl-2-(4-cyclohexyl-piperaz...)
Affinity DataIC50: 1.30nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094156(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2-fluoro-3-trifl...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094182(N-[2-Benzo[1,3]dioxol-4-yl-2-(4-isopropyl-piperazi...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094171(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3-fluoro-2-methy...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469558(CHEMBL4061041)
Affinity DataIC50: 1.46nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC using UDP-3-O-(R-hydroxydecanoyl)-N-acetylglucosamine as substrate preincubated for 30 mins followed by sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094123(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2-chloro-4-fluor...)
Affinity DataIC50: 1.5nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094181(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3-methoxy-phenyl...)
Affinity DataIC50: 1.5nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094154(N-[2-Benzo[1,3]dioxol-4-yl-2-(4-cyclohexyl-piperaz...)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094165(N-(2-Benzo[1,3]dioxol-4-yl-2-[1,4']bipiperidinyl-1...)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094159(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2-fluoro-3-trifl...)
Affinity DataIC50: 1.70nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094168(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3-chloro-4-fluor...)
Affinity DataIC50: 1.70nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094185(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2-chloro-4-fluor...)
Affinity DataIC50: 1.70nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094160(N-(2-Benzo[1,3]dioxol-4-yl-2-[1,4']bipiperidinyl-1...)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094175(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2,3,4-trifluoro-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094144(2-(3,5-Bis-trifluoromethyl-phenyl)-N-[2-(4-cyclohe...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324309(1-{3-[2-(Tetrahydropyran-4-ylamino)pyridin-4-yl][2...)
Affinity DataIC50: 2nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324292(Cyclohexyl-{4-[1-(4-methylpiperazin-1-yl)[2,6]naph...)
Affinity DataIC50: 2nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324294(Cyclohexyl-{4-[1-(4-cyclopropylmethylpiperazin-1-y...)
Affinity DataIC50: 2nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324313(1-{3-[2-(Tetrahydropyran-4-ylamino)pyridin-4-yl][2...)
Affinity DataIC50: 2nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324312(1-{3-[2-(Tetrahydropyran-4-ylamino)pyridin-4-yl][2...)
Affinity DataIC50: 2nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094141(N-(2-[1,4']Bipiperidinyl-1'-yl-2-phenyl-ethyl)-2-(...)
Affinity DataIC50: 2.10nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094119(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataIC50: 2.30nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094140(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2-methoxy-phenyl...)
Affinity DataIC50: 2.40nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094143(2-(3,5-Bis-trifluoromethyl-phenyl)-N-[2-(4-cyclohe...)
Affinity DataIC50: 2.80nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094151(N-(2-Benzo[1,3]dioxol-4-yl-2-[1,4']bipiperidinyl-1...)
Affinity DataIC50: 2.90nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094157(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3-chloro-4-fluor...)
Affinity DataIC50: 2.90nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094139(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3-fluoro-2-methy...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094158(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2,3,5-trichloro-...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324310(1-{3-[2-(Tetrahydropyran-4-ylamino)pyridin-4-yl][2...)
Affinity DataIC50: 3nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324304(1-[3-(2-Cyclohexylaminopyridin-4-yl)[2,6]naphthyri...)
Affinity DataIC50: 3nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324291(Cyclohexyl-{4-[1-((cis-3,5-dimethylpiperazin-1-yl)...)
Affinity DataIC50: 3nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324311(1-{3-[2-(Tetrahydropyran-4-ylamino)pyridin-4-yl][2...)
Affinity DataIC50: 3nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human HDAC1 using rhodamine as substrate after 1 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50249583(CHEMBL4097399)
Affinity DataIC50: 3.13nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC using UDP-3-O-(R-hydroxydecanoyl)-N-acetylglucosamine as substrate preincubated for 30 mins followed by sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetSubstance-P receptor(Human)
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094134(N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3,4-difluoro-phe...)
Affinity DataIC50: 3.30nMAssay Description:Inhibitory activity against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469562(CHEMBL4069725)
Affinity DataIC50: 3.56nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC using UDP-3-O-(R-hydroxydecanoyl)-N-acetylglucosamine as substrate preincubated for 30 mins followed by sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtein kinase C alpha type(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM3033(Indolocarbazole deriv. | 3-{23-methyl-14-oxo-3,13,...)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of PKCalpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50324307({1-[3-(2-Cyclohexylaminopyridin-4-yl)[2,6]naphthyr...)
Affinity DataIC50: 4nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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