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TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003780(CHEMBL435590 | 4-(3-Pyridin-3-yl-propyl)-8-(toluen...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003792(CHEMBL136762 | 8-(4-Fluoro-benzenesulfonylamino)-4...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003784(CHEMBL137402 | 8-(4-Chloro-benzenesulfonylamino)-4...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataIC50: 1nMAssay Description:Concentration required for 50% inhibition of [3H]-CHA binding on rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003803(CHEMBL136738 | 8-(Naphthalene-2-sulfonylamino)-4-(...)
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003801(CHEMBL139372 | 4-(3-Pyridin-3-yl-propyl)-8-(4-trif...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003781(CHEMBL341686 | [5-(4-Chloro-benzenesulfonylamino)-...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003776(CHEMBL65414 | CGS-22652 | 8-(4-Chloro-benzenesulfo...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of thromboxane synthetase in microsomal platelet preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003776(CHEMBL65414 | CGS-22652 | 8-(4-Chloro-benzenesulfo...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003776(CHEMBL65414 | CGS-22652 | 8-(4-Chloro-benzenesulfo...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibition against thromboxane synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003797(CHEMBL63904 | 8-(4-Chloro-benzenesulfonylamino)-4-...)
Affinity DataIC50: 2.60nMAssay Description:In vitro inhibition of thromboxane synthetase in microsomal platelet preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003795(5-[Pyridin-3-yl-(3-trifluoromethyl-phenyl)-methyle...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003798(CHEMBL134580 | 8-(4-Chloro-benzenesulfonylamino)-4...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003799(CHEMBL136934 | 8-(4-Chloro-benzenesulfonylamino)-2...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003800(CHEMBL344457 | 8-(4-Methoxy-benzenesulfonylamino)-...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003796(CHEMBL136371 | 8-(4-Chloro-benzenesulfonylamino)-4...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003797(CHEMBL63904 | 8-(4-Chloro-benzenesulfonylamino)-4-...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50025953(6-Imidazo[1,5-a]pyridin-5-yl-hexanoic acid | CGS-1...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003795(5-[Pyridin-3-yl-(3-trifluoromethyl-phenyl)-methyle...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition against thromboxane synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50046312(8-(4-Chloro-benzenesulfonylamino)-4-[2-(pyridin-3-...)
Affinity DataIC50: 3.5nMAssay Description:In vitro inhibition of thromboxane synthetase in microsomal platelet preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003789(CHEMBL138328 | 8-(4-Methanesulfonyl-benzenesulfony...)
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003794(CHEMBL137505 | 8-(4-Azido-benzenesulfonylamino)-4-...)
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50283051((Z)-7-[(2S,3R,4R)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)
Affinity DataIC50: 4.30nMAssay Description:In vitro inhibition against thromboxane synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50283051((Z)-7-[(2S,3R,4R)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)
Affinity DataIC50: 4.30nMAssay Description:In vitro inhibition against thromboxane synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50046311(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)
Affinity DataIC50: 4.5nMAssay Description:In vitro inhibition of thromboxane synthetase in microsomal platelet preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003787(CHEMBL138743 | 4-Chloro-N-{8-pyridin-3-yl-5-[2-(5H...)
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50046309(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of thromboxane synthetase in microsomal platelet preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50118810(CHEMBL139000 | N6-[(R)-1-Methyl-2-phenylethyl]ado ...)
Affinity DataIC50: 5nMAssay Description:Concentration required for 50% inhibition of [3H]-CHA binding on rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50009552(CHA | CHEMBL45891 | N6-Cyclohexylado (CHA) | 2-[6-...)
Affinity DataIC50: 5nMAssay Description:Concentration required for 50% inhibition of [3H]-CHA binding on rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003790(CHEMBL136880 | Potassium; 8-(4-chloro-benzenesulfo...)
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003804(CHEMBL345105 | 7-(4-Chloro-benzenesulfonylamino)-3...)
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50280267([3-[3-(4-Chloro-benzenesulfonylamino)-propyl]-5-(2...)
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against thromboxane synthase enzyme from human microsomal platelet preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50280268(3-[3-[2-(4-Chloro-benzenesulfonylamino)-ethyl]-5-(...)
Affinity DataIC50: 9nMAssay Description:Inhibitory concentration against thromboxane synthase enzyme from human microsomal platelet preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003793(CHEMBL134686 | 8-(4-Chloro-benzenesulfonylamino)-4...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50283046((Z)-7-[(2S,3S,4S)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50283042((Z)-7-[(2S,3S,4R)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283049(GR 32191 | CHEMBL65030 | GR-32191 | (Z)-7-[(1R,2R,...)
Affinity DataIC50: 12nMAssay Description:In vitro thromboxane receptor antagonist activity was determined by inhibition of U-46619 induced aggregation of washed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50046310(8-(4-Chloro-benzenesulfonylamino)-4-[2-(pyridin-3-...)
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of thromboxane synthetase in microsomal platelet preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50283046((Z)-7-[(2S,3S,4S)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50283046((Z)-7-[(2S,3S,4S)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a/A2b(Rat)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50009535(CHEMBL314313 | 2-[6-Amino-2-(2-cyclohex-1-enyl-eth...)
Affinity DataIC50: 13nMAssay Description:Concentration required for 50% inhibition of [3H]NECA binding on rat brain adenosine A2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50280260(7-{4-[3-(4-Chloro-benzenesulfonylamino)-propyl]-py...)
Affinity DataIC50: 15nMAssay Description:Inhibitory concentration against thromboxane synthase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50280264(3-[5-[2-(4-Chloro-benzenesulfonylamino)-ethyl]-2-(...)
Affinity DataIC50: 15nMAssay Description:Inhibitory concentration against thromboxane synthase enzyme from human microsomal platelet preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAdenosine receptor A2a/A2b(Rat)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 15nMAssay Description:Concentration required for 50% inhibition of [3H]NECA binding on rat brain adenosine A2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 16nMAssay Description:Concentration required for 50% inhibition of [3H]-CHA binding on rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50283051((Z)-7-[(2S,3R,4R)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)
Affinity DataIC50: 17nMAssay Description:In vitro inhibition against thromboxane synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a/A2b(Rat)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50009543(CHEMBL2374391 | 2-{6-Amino-2-[2-(5,6,7,8-tetrahydr...)
Affinity DataIC50: 17nMAssay Description:Concentration required for 50% inhibition of [3H]NECA binding on rat brain adenosine A2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50003791(CHEMBL343535 | [5-(4-Chloro-benzenesulfonylamino)-...)
Affinity DataIC50: 18nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283047((Z)-7-[(2S,3S,4S)-4-(Biphenyl-4-ylmethoxy)-1,1-dio...)
Affinity DataIC50: 18nMAssay Description:In vitro thromboxane receptor antagonist activity was determined by inhibition of U-46619 induced aggregation of washed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50003776(CHEMBL65414 | CGS-22652 | 8-(4-Chloro-benzenesulfo...)
Affinity DataIC50: 18nMAssay Description:In vitro thromboxane receptor antagonist activity was determined by inhibition of U-46619 induced aggregation of washed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

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